Affinity DataKi: 740nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
Affinity DataKi: 744nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
Affinity DataKi: 7.00E+4nMAssay Description:Inhibition of acid sphingomyelinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 8.50E+4nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
Affinity DataKi: 1.39E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
Affinity DataKi: 1.55E+5nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
Affinity DataKi: 1.74E+5nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced platelet aggregation in human whole bloodMore data for this Ligand-Target Pair
Affinity DataKi: 3.54E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
Affinity DataKi: 3.90E+5nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced platelet aggregation in human whole bloodMore data for this Ligand-Target Pair
Affinity DataKi: 5.40E+5nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
Affinity DataKi: 5.88E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
Affinity DataKi: 9.55E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
Affinity DataKi: 1.42E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+6nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
Affinity DataKi: 4.74E+6nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+6nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced platelet aggregation in human whole bloodMore data for this Ligand-Target Pair
Affinity DataKi: 6.22E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
Affinity DataKi: 6.38E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+7nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+7nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of acid sphingomyelinase (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human RIPK1 incubated for 40 min in presence of ATP by ADP-Glo luminescence kinase assayMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 92nMAssay Description:Inhibition of human RIPK1 incubated for 40 min in presence of ATP by ADP-Glo luminescence kinase assayMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 186nMAssay Description:Inhibition of human RIPK1 incubated for 40 min in presence of ATP by ADP-Glo luminescence kinase assayMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 298nMAssay Description:Inhibition of human RIPK1 incubated for 40 min in presence of ATP by ADP-Glo luminescence kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of human Huh7 cell derived acid sphingomyelinase using NBD-sphingomyelin as substrate after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of human Huh7 cell derived acid sphingomyelinase using NBD-sphingomyelin as substrate after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition of human Huh7 cell derived acid sphingomyelinase using NBD-sphingomyelin as substrate after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition of recombinant human acid sphingomyelinase (His62 to Pro628 residues) using NBD-sphingomyelin as substrate after 30 mins by fluorescence b...More data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibition of human Huh7 cell derived acid sphingomyelinase using NBD-sphingomyelin as substrate after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphoglycerate mutase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of recombinant His-tagged PGAM1 (unknown origin) expressed in Escherichia coli BL21 using 3-PG as substrate in presence of ADP by Kinase-G...More data for this Ligand-Target Pair
TargetPhosphoglycerate mutase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of PGAM1 (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 624nMAssay Description:Inhibition of human RIPK1 incubated for 40 min in presence of ATP by ADP-Glo luminescence kinase assayMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 693nMAssay Description:Inhibition of human RIPK1 incubated for 40 min in presence of ATP by ADP-Glo luminescence kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:Inhibition of human Huh7 cell derived acid sphingomyelinase using NBD-sphingomyelin as substrate after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 890nMAssay Description:Inhibition of recombinant human acid sphingomyelinase (His62 to Pro628 residues) using NBD-sphingomyelin as substrate after 30 mins by fluorescence b...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of human RIPK1 incubated for 40 min in presence of ATP by ADP-Glo luminescence kinase assayMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of human RIPK1 incubated for 40 min in presence of ATP by ADP-Glo luminescence kinase assayMore data for this Ligand-Target Pair
TargetPhosphoglycerate mutase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of PGAM1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.73E+3nMAssay Description:Inhibition of human Huh7 cell derived acid sphingomyelinase using NBD-sphingomyelin as substrate after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphoglycerate mutase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of PGAM1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.96E+3nMAssay Description:Inhibition of human Huh7 cell derived acid sphingomyelinase using NBD-sphingomyelin as substrate after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of human Huh7 cell derived acid sphingomyelinase using NBD-sphingomyelin as substrate after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human acid sphingomyelinase (His62 to Pro628 residues) using NBD-sphingomyelin as substrate after 30 mins by fluorescence b...More data for this Ligand-Target Pair
TargetPhosphoglycerate mutase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of PGAM1 (unknown origin)More data for this Ligand-Target Pair
TargetPhosphoglycerate mutase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of PGAM1 (unknown origin)More data for this Ligand-Target Pair
TargetPhosphoglycerate mutase 1(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of PGAM1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of acid sphingomyelinase (unknown origin)More data for this Ligand-Target Pair