TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]DTG from S1R in P2 fraction of Hartley guinea pig whole brain after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 111nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 125nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 131nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 135nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 167nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 171nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 178nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 211nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 286nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 301nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 340nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 462nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataKi: 606nMAssay Description:Displacement of [3H](+)-pentazocine from S1R in guinea pig brain cortex membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 704nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 749nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 802nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Displacement of [3H]-DTG from S2R in rat liver membranes after 120 mins by scintillation counting assayMore data for this Ligand-Target Pair