TargetCalcium/calmodulin-dependent protein kinase type II subunit beta(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of CAMK2b (unknown origin)More data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of RSK1 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of JAK3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inhibition of CHK1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 1(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.367nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.370nMAssay Description:Inhibition of PKCalpha (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.450nMAssay Description:Inhibition of PDGFRalpha (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.450nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
TargetMisshapen-like kinase 1(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.470nMAssay Description:Inhibition of MINK1 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.473nMAssay Description:Inhibition of LYN (unknown origin)More data for this Ligand-Target Pair
TargetPhosphorylase b kinase gamma catalytic chain, liver/testis isoform(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.490nMAssay Description:Inhibition of PHKg2 (unknown origin)More data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.640nMAssay Description:Inhibition of ROCK1 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.720nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin)More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 0.860nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of LCK (unknown origin) after 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of TRKA (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of LCK (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of CDK1/cyclin B (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of RET (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G1/S-specific cyclin- 1(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of CDK1/cyclin E (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of c-SRC (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of VEGFR3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Inhibition of PAK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of AKT1 (unknown origin)More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Inhibition of FMS (unknown origin) after 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 3(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Inhibition of STK3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of CHK2 (unknown origin)More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 5.40nMAssay Description:Inhibition of GSK3beta (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of LCK (unknown origin) after 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 6.20nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of LCK (unknown origin) after 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 7.30nMAssay Description:Inhibition of MAPK15 (unknown origin)More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat cerebral cortex membranes after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 8.20nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Inhibition of FMS (unknown origin) after 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 9.30nMAssay Description:Inhibition of FGFR3 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat cerebral cortex membranes after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetDeath-associated protein kinase 1(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of FMS (unknown origin) after 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
TargetInsulin receptor(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of IR (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of MAPK14 (unknown origin)More data for this Ligand-Target Pair
TargetEphrin type-A receptor 3(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of EPHA3 (unknown origin)More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of FMS (unknown origin) after 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of LCK (unknown origin) after 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Korea Institute of Science & Technology (Kist)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition concentration against human adenosine kinaseMore data for this Ligand-Target Pair