Compile Data Set for Download or QSAR
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Found 10 with Last Name = 'kuppast' and Initial = 'b'
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50074501(Butyl-ethyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-ph...)
Affinity DataIC50:  19nMAssay Description:Displacement of [125I]Tyr0sauvagine from human CRF1 receptor expressed in HEK293 cell membrane after 120 mins by gamma scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50074501(Butyl-ethyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-ph...)
Affinity DataIC50:  19nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50276840(CHEMBL4160471)
Affinity DataIC50:  170nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50003912(CHEMBL3235706)
Affinity DataIC50:  245nMAssay Description:Displacement of [125I]Tyr0sauvagine from human CRF1 receptor expressed in HEK293 cell membrane after 120 mins by gamma scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50003909(CHEMBL3235700)
Affinity DataIC50:  275nMAssay Description:Displacement of [125I]Tyr0sauvagine from human CRF1 receptor expressed in HEK293 cell membrane after 120 mins by gamma scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50276841(CHEMBL4161963)
Affinity DataIC50:  447nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50003910(CHEMBL3235703)
Affinity DataIC50:  537nMAssay Description:Displacement of [125I]Tyr0sauvagine from human CRF1 receptor expressed in HEK293 cell membrane after 120 mins by gamma scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50003911(CHEMBL3235705)
Affinity DataIC50:  589nMAssay Description:Displacement of [125I]Tyr0sauvagine from human CRF1 receptor expressed in HEK293 cell membrane after 120 mins by gamma scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50276839(CHEMBL4170184)
Affinity DataIC50:  891nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50276840(CHEMBL4160471)
Affinity DataEC50:  1.10nMAssay Description:Antagonist activity at human CRFR1 expressed in HEK293 cells assessed as inhibition of sauvagine-induced cAMP accumulation by measuring sauvagine EC5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed