Affinity DataKi: 1.5nMAssay Description:Binding affinity of the compound for NK-1 receptor was determined in a radioligand binding assay using IM9 human lymphoblastoma cell line.More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity of the compound for NK-3 receptor was determined in vitro using isolated rat portal vein.More data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Binding affinity of the compound for NK-2 receptor was determined in vitro using isolated rabbit pulmonary artery.More data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Binding affinity of the compound for NK-3 receptor was determined in vitro using isolated rat portal vein.More data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Binding affinity of the compound for NK-2 receptor was determined in vitro using isolated rabbit pulmonary artery.More data for this Ligand-Target Pair
Affinity DataKi: 8nM ΔG°: -43.0kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Antagonistic potency for NK-1 receptor was determined in a radioligand binding assay, using IM9 human lymphoblastoma cell line.More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity of the compound for NK-1 receptor was determined in vitro using isolated rabbit vena cava.More data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Antagonistic potency for NK-2 receptor was determined in vitro, using isolated rabbit pulmonary artery.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18.4nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataKi: 54.2nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
Affinity DataKi: 254nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataKi: 378nM ΔG°: -34.1kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Affinity DataKi: 515nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: 579nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: 583nM ΔG°: -33.1kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Affinity DataKi: 618nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
Affinity DataKi: 695nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: 718nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: 947nM ΔG°: -32.0kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Affinity DataKi: 947nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: 969nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+3nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.93E+3nM ΔG°: -30.3kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Antagonistic potency for NK-2 receptor was determined in vitro, using isolated rabbit pulmonary artery.More data for this Ligand-Target Pair
Affinity DataKi: 3.81E+3nM ΔG°: -28.8kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Affinity DataKi: 4.20E+3nMAssay Description:Binding affinity of the compound for NK-2 receptor was determined in vitro using isolated rabbit pulmonary artery.More data for this Ligand-Target Pair
Affinity DataKi: 4.39E+3nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: 6.69E+3nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
![](/img/powered_by_small.gif)