Report error Found 144 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM28681'
Affinity DataEC50: 40nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase activity w...More data for this Ligand-Target Pair
Affinity DataKd: 14.8nM EC50: 3.80nMpH: 7.5 T: 2°CAssay Description:Kd values were obtained by incubating His-PPARgamma-LBD with biotinylated peptide, europium-labeled anti-histidine antibody, and allophycocyanin-labe...More data for this Ligand-Target Pair
Affinity DataEC50: 82nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Agonistic activity was determined in COS1 cells transfected with GAL 4-PPAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Maximal reporter activity against human Peroxisome proliferator activated receptor gamma Gal4 chimeric in transiently transfected CV-1 cells by funct...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:In vitro transactivation of human peroxisome proliferator activated receptor gamma measured in PPAR-GAL4 chimeric COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 89nMAssay Description:Activation of peroxisome proliferator activated receptor gamma measured by induction of 50% of maximum alkaline phosphatase activity, transfection as...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxo Wellcome Research and Development
Curated by ChEMBL
Glaxo Wellcome Research and Development
Curated by ChEMBL
Affinity DataEC50: 60nMAssay Description:In vitro transcriptional activation of Peroxisome proliferator activated receptor gamma (PPAR) expressed in CV-1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxo Wellcome Research and Development
Curated by ChEMBL
Glaxo Wellcome Research and Development
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Agonist activity for murine PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Agonist activity for Human PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at human PPARgamma receptor expressed in african green monkey COS1 cells co-transfected with fused yeast Gal4-DBD by transactivation...More data for this Ligand-Target Pair
Affinity DataEC50: 657nMAssay Description:Binding affinity at human PPAR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:In vitro transactivation using receptor transactivation assay against hPPAR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:In vitro activation of human peroxisome proliferator activated receptor gamma (PPAR gamma)More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:In vitro agonist activity tested for transactivation in human PPAR gamma-Gal4 chimeric COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:In vitro transactivation of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Transcriptional activation by human PPAR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:In vitro potency of PPAR gene activation against human PPAR gamma receptor using chimeric Gal4-hPPAR transactivation assay (TA)More data for this Ligand-Target Pair
Affinity DataEC50: 2.88E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Effective concentration against human peroxisome proliferator activated receptor gamma in Gal4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 268nMAssay Description:Mean effective concentration against human peroxisome proliferator-activated receptor gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Effective concentration against human Peroxisome proliferator activated receptor gamma in Gal4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 140nMAssay Description:Effective concentration against human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Maximal intrinsic response against peroxisome proliferator activated receptor gamma transactivationMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 39nMAssay Description:Effective concentration against human PPARgamma expressed in HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Effective agonist concentration for human PPAR gamma Gal4 construct in transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 308nMAssay Description:Transactivation of human PPARgamma in CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Activity at human PPAR gamma transfected in NIH3T3 cells by luciferase activity assayMore data for this Ligand-Target Pair
Affinity DataEC50: 308nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 308nMAssay Description:Agonist activity at PPARgamma in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at human PPARgamma by transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Agonist activity at PPARgamma receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 310nMAssay Description:Activity at human adipose tissue PPAR gamma expressed in HEK293 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Agonist activity at human PPARgamma in CV1 cells by GAL4 transactivation assay after 24 hrsMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Agonist activity at human PPARgamma by transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Agonist activity at human PPARgamma expressed in NIH3T3 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 308nMAssay Description:Agonist activity at human PPARgamma expressed in CV1 cells by receptor transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 33nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV-1 co-transfected with GAL4 by by dual-glo luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at PPARgamma expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assay relative to con...More data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Agonist activity at PPARgamma ligand binding domain expressed in human HeLa cells co-transfected with Gal4-DBD assessed as transcriptional activation...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at human recombinant PPARgamma expressed in COS1 cells co-expressing GAL4 assessed as transcriptional activity after 48 hrs by lucif...More data for this Ligand-Target Pair
Affinity DataEC50: 450nMAssay Description:Agonist activity at human PPARgamma expressed in BHK21 cells assessed as SEAP activity by luciferase reporter transactivation assayMore data for this Ligand-Target Pair
