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Found 49 with Last Name = 'espinosa-bustos' and Initial = 'c'
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510725(CHEMBL4560144)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510722(CHEMBL4572026)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510721(CHEMBL4568106)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510717(CHEMBL4446112)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510715(CHEMBL4544939)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510720(CHEMBL4476179)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50177729(Aplysamine-1 | CHEMBL380697 | aplysamine)
Affinity DataKi:  30nMAssay Description:Inhibition of histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510726(CHEMBL4451014)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510714(CHEMBL4526393)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510719(CHEMBL4436457)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510724(CHEMBL4560119)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510718(CHEMBL4573388)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50462996(CHEMBL4242249)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50462998(CHEMBL4241911)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510723(CHEMBL4439125)
Affinity DataKi:  317nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510713(CHEMBL4476221)
Affinity DataKi:  374nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50462997(CHEMBL4239928)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510716(CHEMBL4566980)
Affinity DataKi:  848nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50462999(CHEMBL4242697)
Affinity DataKi:  1.07E+3nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510715(CHEMBL4544939)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510725(CHEMBL4560144)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510726(CHEMBL4451014)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510722(CHEMBL4572026)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510724(CHEMBL4560119)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510721(CHEMBL4568106)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510720(CHEMBL4476179)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510719(CHEMBL4436457)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510718(CHEMBL4573388)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510717(CHEMBL4446112)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510716(CHEMBL4566980)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510723(CHEMBL4439125)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510714(CHEMBL4526393)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510713(CHEMBL4476221)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153275((E)-3-(4-Bromo-2,5-dimethoxyphenyl)-1-(2-hydroxy-5...)
Affinity DataIC50:  2.80E+3nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153273((E)-3-(4-Bromo-2,5-dimethoxyphenyl)-1-(2-hydroxy-6...)
Affinity DataIC50:  6.10E+3nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153274((E)-3-(2,3-Dimethoxyphenyl)-1-(2-hydroxy-5-methoxy...)
Affinity DataIC50:  6.80E+3nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153272((E)-3-(2,5-Dimethoxyphenyl)-1-(2-hydroxy-6-methoxy...)
Affinity DataIC50:  1.09E+4nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153278((Z)-2-(2,3-Dimethoxybenzylidene)-5-methoxybenzofur...)
Affinity DataIC50:  1.16E+4nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153279((Z)-2-(4-Bromo-2,5-dimethoxybenzylidene)-5-methoxy...)
Affinity DataIC50:  1.35E+4nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153276((Z)-2-(2,5-Dimethoxybenzylidene)-4-methoxybenzofur...)
Affinity DataIC50:  1.78E+4nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153277((Z)-2-(4-Bromo-2,5-dimethoxybenzylidene)-4-methoxy...)
Affinity DataIC50:  2.63E+4nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153272((E)-3-(2,5-Dimethoxyphenyl)-1-(2-hydroxy-6-methoxy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153275((E)-3-(4-Bromo-2,5-dimethoxyphenyl)-1-(2-hydroxy-5...)
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153279((Z)-2-(4-Bromo-2,5-dimethoxybenzylidene)-5-methoxy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153278((Z)-2-(2,3-Dimethoxybenzylidene)-5-methoxybenzofur...)
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153274((E)-3-(2,3-Dimethoxyphenyl)-1-(2-hydroxy-5-methoxy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153273((E)-3-(4-Bromo-2,5-dimethoxyphenyl)-1-(2-hydroxy-6...)
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153277((Z)-2-(4-Bromo-2,5-dimethoxybenzylidene)-4-methoxy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile

LigandPNGBDBM153276((Z)-2-(2,5-Dimethoxybenzylidene)-4-methoxybenzofur...)
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed