TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 121nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 148nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 317nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 374nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 848nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 1.07E+3nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: 2.80E+3nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: 6.10E+3nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: 6.80E+3nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: 1.09E+4nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: 1.16E+4nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: 1.35E+4nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: 1.78E+4nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: 2.63E+4nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Pontificia Universidad Catolica De Chile
Pontificia Universidad Catolica De Chile
Affinity DataIC50: >1.00E+5nMAssay Description:Briefly, a crude rat brain mitochondrial suspension (male SpragueżDawley rats weighing 180ż220 g, killed by decapitation) was used as protein source....More data for this Ligand-Target Pair
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