Affinity DataKi: 0.380nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Receptor binding affinity against Sigma-1 receptor from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.880nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Receptor binding affinity against Sigma-1 receptor from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.02nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.24nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Receptor binding affinity against Sigma receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10.5nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Receptor binding affinity against Sigma receptorMore data for this Ligand-Target Pair
Affinity DataKi: <17.7nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseMore data for this Ligand-Target Pair
Affinity DataKi: <21nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseMore data for this Ligand-Target Pair
Affinity DataKi: 24.3nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition of Staphylococcus aureus DNA topoisomerase 4More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Inhibition of Staphylococcus aureus DNA topoisomerase 4More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:In vitro for binding affinity at sigma-1 receptor by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKd: 3.10nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Affinity DataKd: <3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
Affinity DataKd: 7.20E+3nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Affinity DataKd: 1.60E+3nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Affinity DataKd: 8.90nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Affinity DataKd: 970nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Affinity DataKd: 250nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Affinity DataKd: 210nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Affinity DataKd: 52nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Stanford University
Curated by ChEMBL
Stanford University
Curated by ChEMBL
Affinity DataKd: 4.5nMAssay Description:Inhibition of wild-type human partial length KIT (I571 to D952 residues) expressed in bacterial expression system by ATP-site competition binding ass...More data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
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