Affinity DataKi: 5nMAssay Description:Mixed inhibition of Electrophorus electricus acetylcholinesterase using acetylcholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Non-competitive inhibition of rat liver mitochondrial MAO-B using phenylethylamine as substrate by Line-Weaver Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 20.2nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of AChE (unknown orign) by Lineweaver-Burke plotMore data for this Ligand-Target Pair
Affinity DataKi: 38.9nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 41.9nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 61.3nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Mixed-type inhibition of electric eel AChE using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 149nMAssay Description:Mixed type inhibition of Electrophorus electricus AchE using acetylthiocholine as substrate by Line-Weaver Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 157nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 621nMAssay Description:Mixed-type inhibition of Electrophorus electricus AChE assessed as hydrolysis of acetylthiocholine by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataKi: 7.10E+3nMAssay Description:Competitive inhibition of equine serum BChE using acetylthiocholine as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Affinity DataIC50: 0.0250nMAssay Description:Inhibition of mitochondrial MAO-B in rat liver homogenates using [14C]-phenylethylamine as substrate preincubated for 30 mins by liquid scintillation...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 0.790nMAssay Description:Inhibition of mitochondrial MAO-A in rat liver homogenates using [14C]-(5-hydroxy-triptamine) as substrate preincubated for 30 mins by liquid scintil...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Inhibition of rat liver mitochondrial MAO-A using [14C]-5-hydroxytryptamine after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Inhibition of horse serum BuChE by Ellman's methodMore data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Inhibition of horse serum BChE after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Inhibition of horse serum butrylcholinesterase preincubated with compound for 10 mins using butrylcholine iodide as substrate after 15 mins by spectr...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Inhibition of equine serum BuChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 6.70nMAssay Description:Inhibition of rat liver mitochondrial MAO-A using [14C]-5-hydroxytryptamine after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins measured after 15 mins of substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase preincubated with compound for 10 mins using acetylcholine iodide as substrate after 15 m...More data for this Ligand-Target Pair
Affinity DataIC50: 8.20nMAssay Description:Inhibition of AChE in human erythrocytes by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of rat liver mitochondrial MAO-A using [14C]-5-hydroxytryptamine after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 13.4nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase preincubated with compound for 10 mins using acetylcholine iodide as substrate after 15 m...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase preincubated with compound for 10 mins using acetylcholine iodide as substrate after 15 m...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase preincubated with compound for 10 mins using acetylcholine iodide as substrate after 15 m...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of mitochondrial MAO-B in rat liver homogenates using [14C]-phenylethylamine as substrate preincubated for 30 mins by liquid scintillation...More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase preincubated with compound for 10 mins using acetylcholine iodide as substrate after 15 m...More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase preincubated with compound for 10 mins using acetylcholine iodide as substrate after 15 m...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of electric eel AChE after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by Ellman'...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase preincubated with compound for 10 mins using acetylcholine iodide as substrate after 15 m...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Displacement of propidium iodide from AChE in bovine erythrocytes after 15 mins by fluorescence plate readerMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase preincubated with compound for 10 mins using acetylcholine iodide as substrate after 15 m...More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair