Affinity DataIC50: 0.0790nMAssay Description:Tested for binding affinity of compound against [125I]NKA binding to neurokinin-2 (NK-2) receptor in hamster urinary bladderMore data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 141nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 151nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Tested for binding affinity against [125I]BH-SP binding to neurokinin-1 (NK-1) receptor in human IM-9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.59E+3nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Binding affinity towards Tachykinin receptor 3 using [125I]-[Mephe7] NKB as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.09E+3nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity towards Tachykinin receptor 3 using [125I]-[Mephe7] NKB as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [3H]senktide to Tachykinin receptor 3 in the guinea pig cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Tested for binding affinity against [125I]BH-SP binding to neurokinin-1 (NK-1) receptor in human IM-9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.72E+3nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+3nMAssay Description:Binding affinity towards Tachykinin receptor 3 using [125I]-[Mephe7] NKB as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+3nMAssay Description:Tested for binding affinity of compound against [125I]NKA binding to neurokinin-2 (NK-2) receptor in hamster urinary bladderMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+3nMAssay Description:Binding affinity towards Tachykinin receptor 2 using [125I]iodohistidyl-NKA (0.1 nM)) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Tested for binding affinity against [125I]BH-SP binding to neurokinin-1 (NK-1) receptor in human IM-9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.24E+3nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 7.41E+3nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 9.30E+3nMAssay Description:Tested for binding affinity against [125I]BH-SP binding to neurokinin-1 (NK-1) receptor in human IM-9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30E+3nMAssay Description:Binding affinity towards Tachykinin receptor 3 using [125I]-[Mephe7] NKB as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+3nMAssay Description:Binding affinity towards Tachykinin receptor 3 using [125I]-[Mephe7] NKB as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Tachykinin receptor 2 using [125I]iodohistidyl-NKA (0.1 nM)) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Tested for binding affinity of compound against [125I][MePhe]-NKB binding to Tachykinin receptor 3 in stably expressed CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Tachykinin receptor 2 using [125I]iodohistidyl-NKA (0.1 nM)) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.98E+4nMAssay Description:Binding affinity towards Tachykinin receptor 2 using [125I]iodohistidyl-NKA (0.1 nM)) as radioligandMore data for this Ligand-Target Pair