Affinity DataKi: 5.30E+3nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 7.60E+3nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.08E+4nMAssay Description:Displacement of fluorescent-tagged BH3 domain of Bak from Bcl-xL by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.41E+4nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.78E+4nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of fluorescent-tagged BH3 domain of Bak from Bcl-xL by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Laboratoire Des M£Canismes Mol£Culaires Des Communications Cellulaires (Cnrs Upr 9023)
Curated by ChEMBL
Laboratoire Des M£Canismes Mol£Culaires Des Communications Cellulaires (Cnrs Upr 9023)
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Compound was tested in vitro for inhibition of tubulin polymerization.More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles (Icsn)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair