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Found 266 with Last Name = 'koga' and Initial = 'h'
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50101813(CHEBI:31399 | Cilnidipine)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of voltage-dependent L-type calcium channel in rat thoracic aorta ring assessed as effect on high K+ induced contraction by Magnus methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50101813(CHEBI:31399 | Cilnidipine)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of Voltage-dependent L-type calcium channel in rat thoracic aorta ringMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50101813(CHEBI:31399 | Cilnidipine)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421355(CHEMBL289955)
Affinity DataIC50:  1.80nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421358(CHEMBL45141)
Affinity DataIC50:  1.90nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421357(CHEMBL297168)
Affinity DataIC50:  2.30nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421355(CHEMBL289955)
Affinity DataIC50:  2.5nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  2.60nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475660(CHEMBL201566)
Affinity DataIC50:  2.80nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421354(CHEMBL26966)
Affinity DataIC50:  3.20nMAssay Description:Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50More data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421354(CHEMBL26966)
Affinity DataIC50:  3.20nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421356(CHEMBL43313)
Affinity DataIC50:  3.5nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475658(CHEMBL201984)
Affinity DataIC50:  3.70nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421349(CHEMBL265495)
Affinity DataIC50:  3.80nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421349(CHEMBL265495)
Affinity DataIC50:  3.80nMAssay Description:Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50More data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421356(CHEMBL43313)
Affinity DataIC50:  3.80nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421357(CHEMBL297168)
Affinity DataIC50:  3.90nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [588-1127,Y768C]/[588-1147,Y768C](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  4nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1127,Y768C]/[588-1147,Y768C](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  4nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM5052(5-bromo-N-[(2Z)-4-chloro-3-methyl-5-(propan-2-yl)-...)
Affinity DataIC50:  4.30nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475653(CHEMBL382528)
Affinity DataIC50:  5.80nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421351(CHEMBL27424)
Affinity DataIC50:  6nMAssay Description:Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50More data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421351(CHEMBL27424)
Affinity DataIC50:  6nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421349(CHEMBL265495)
Affinity DataIC50:  6.5nMpH: 2.5 T: 2°CAssay Description:Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution fo...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421349(CHEMBL265495)
Affinity DataIC50:  6.5nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
In DepthDetails Article
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475650(CHEMBL203041)
Affinity DataIC50:  6.80nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  6.90nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  6.90nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50479255(CHEMBL453084)
Affinity DataIC50:  7nMAssay Description:Inhibition of voltage-dependent L-type calcium channel in rat thoracic aorta ring assessed as effect on high K+ induced contraction by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421351(CHEMBL27424)
Affinity DataIC50:  7.90nMpH: 2.5 T: 2°CAssay Description:Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution fo...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421351(CHEMBL27424)
Affinity DataIC50:  7.90nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421350(CHEMBL27419)
Affinity DataIC50:  8.90nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421350(CHEMBL27419)
Affinity DataIC50:  8.90nMpH: 2.5 T: 2°CAssay Description:Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution fo...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421350(CHEMBL27419)
Affinity DataIC50:  8.90nMpH: 2.5 T: 2°CAssay Description:Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution fo...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM5054(5-Chloro-N-(4-chloro-5-isopropyl-3-methyl-1,3-thia...)
Affinity DataIC50:  9nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475663(CHEMBL202464)
Affinity DataIC50:  9nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421350(CHEMBL27419)
Affinity DataIC50:  9.10nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM5051(5-Chloro-N-(4-chloro-5-isopropyl-3-methyl-13-thiaz...)
Affinity DataIC50:  9.40nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM5055(N-(4-Chloro-5-isopropyl-3-methyl-1,3-thiazol-2(3H)...)
Affinity DataIC50:  9.5nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475664(CHEMBL369934)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM5048(5-Chloro-2-cyano-N-(5-isopropyl-3,4-dimethyl-1,3-t...)
Affinity DataIC50:  11nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1127,Y768C]/[588-1147,Y768C](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM5041(N-(5-tert-Butyl-3,4-dimethyl-1,3-thiazol-2(3H)-yli...)
Affinity DataIC50:  11nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM5053(2,5-dicyano-N-[(2Z)-3,4-dimethyl-5-(propan-2-yl)-2...)
Affinity DataIC50:  12nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475672(CHEMBL201057)
Affinity DataIC50:  13nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1127,Y768C]/[588-1147,Y768C](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM5052(5-bromo-N-[(2Z)-4-chloro-3-methyl-5-(propan-2-yl)-...)
Affinity DataIC50:  13nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475662(CHEMBL201860)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical

LigandPNGBDBM5050(5-Bromo-2-cyano-N-(5-isopropyl-3,4-dimethyl-1,3-th...)
Affinity DataIC50:  18nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475669(CHEMBL382072)
Affinity DataIC50:  20nMAssay Description:Inhibition of voltage-dependent L-type calcium channel in rat thoracic aorta ring assessed as effect on high K+ induced contraction by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475669(CHEMBL382072)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475656(CHEMBL201306)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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