BindingDB PrimarySearch_ki

Found 81 with Last Name = 'jerchel-furau' and Initial = 'i'

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610147(CHEMBL5289955)

IC50: 2nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610163(CHEMBL5267263)

IC50: 4.20nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50266373(2-chloro-5-nitro-N-(pyridin-4-yl)benzamide | CHEMB...)

IC50: 4.70nMAssay Description:Inverse agonist activity at human PPARgamma expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for...More data for this Ligand-Target Pair

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3D Structure (crystal)

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610165(CHEMBL5273393)

IC50: 4.80nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610166(CHEMBL5282503)

IC50: 5nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610163(CHEMBL5267263)

IC50: 6.10nMAssay Description:Inverse agonist activity at human PPARgamma expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610161(CHEMBL5281842)

IC50: 6.60nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610152(CHEMBL5268912)

IC50: 7.40nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610167(CHEMBL5271038)

IC50: 8.30nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Mus musculus)TBA

PNG

BDBM50610163(CHEMBL5267263)

IC50: 8.70nMAssay Description:Inverse agonist activity at PPARgamma in mouse 3T3-L1 adipocytes assessed as inhibition of adipogenesis by measuring lipid droplet staining by BODIPY...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM161150(US9051265, 58 | US9051265, 98)

IC50: 12nMAssay Description:Inverse agonist activity at human PPARgamma expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for...More data for this Ligand-Target Pair

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3D Structure (crystal)

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610167(CHEMBL5271038)

IC50: 14nMAssay Description:Inverse agonist activity at human PPARgamma expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610164(CHEMBL5272194)

IC50: 14nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610162(CHEMBL5286386)

IC50: 15nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Mus musculus)TBA

PNG

BDBM50610167(CHEMBL5271038)

IC50: 24nMAssay Description:Inverse agonist activity at PPARgamma in mouse 3T3-L1 adipocytes assessed as inhibition of adipogenesis by measuring lipid droplet staining by BODIPY...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610162(CHEMBL5286386)

IC50: 28nMAssay Description:Inverse agonist activity at human PPARgamma expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610159(CHEMBL5285688)

IC50: 38nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610158(CHEMBL5291018)

IC50: 54nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Mus musculus)TBA

PNG

BDBM50610162(CHEMBL5286386)

IC50: 73nMAssay Description:Inverse agonist activity at PPARgamma in mouse 3T3-L1 adipocytes assessed as inhibition of adipogenesis by measuring lipid droplet staining by BODIPY...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610160(CHEMBL5277957)

IC50: 91nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610148(CHEMBL5287868)

IC50: 94nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Mus musculus)TBA

PNG

BDBM50591456(CHEMBL5207130)

IC50: 148nMAssay Description:Inverse agonist activity at PPARgamma in mouse 3T3-L1 adipocytes assessed as inhibition of adipogenesis by measuring lipid droplet staining by BODIPY...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610145(CHEMBL5283176)

IC50: 183nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor alpha(Homo sapiens (Human))TBA

PNG

BDBM161150(US9051265, 58 | US9051265, 98)

IC50: 935nMAssay Description:Agonist activity at human PPARalpha expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional activation preincubated for 6 hrs f...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610154(CHEMBL5288593)

IC50: 1.04E+3nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610143(CHEMBL5278668)

IC50: 1.12E+3nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610151(CHEMBL5282181)

IC50: 2.20E+3nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor alpha(Homo sapiens (Human))TBA

PNG

BDBM50266373(2-chloro-5-nitro-N-(pyridin-4-yl)benzamide | CHEMB...)

IC50: 2.95E+3nMAssay Description:Agonist activity at human PPARalpha expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional activation preincubated for 6 hrs f...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610149(CHEMBL5272116)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Thyroid hormone receptor beta(Homo sapiens (Human))TBA

PNG

BDBM50610163(CHEMBL5267263)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human THRB expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for 6 hr...More data for this Ligand-Target Pair

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Thyroid hormone receptor beta(Homo sapiens (Human))TBA

PNG

BDBM50610162(CHEMBL5286386)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human THRB expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for 6 hr...More data for this Ligand-Target Pair

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Thyroid hormone receptor alpha(Homo sapiens (Human))TBA

PNG

BDBM50610167(CHEMBL5271038)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human THRA expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for 6 hr...More data for this Ligand-Target Pair

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Thyroid hormone receptor alpha(Homo sapiens (Human))TBA

PNG

BDBM50610163(CHEMBL5267263)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human THRA expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for 6 hr...More data for this Ligand-Target Pair

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Thyroid hormone receptor alpha(Homo sapiens (Human))TBA

PNG

BDBM50610162(CHEMBL5286386)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human THRA expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for 6 hr...More data for this Ligand-Target Pair

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Bile acid receptor(Homo sapiens (Human))TBA

PNG

BDBM50610167(CHEMBL5271038)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human FXR expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for 6 hrs...More data for this Ligand-Target Pair

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Bile acid receptor(Homo sapiens (Human))TBA

PNG

BDBM50610163(CHEMBL5267263)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human FXR expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for 6 hrs...More data for this Ligand-Target Pair

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Bile acid receptor(Homo sapiens (Human))TBA

PNG

BDBM50610162(CHEMBL5286386)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human FXR expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for 6 hrs...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor delta(Homo sapiens (Human))TBA

PNG

BDBM50266373(2-chloro-5-nitro-N-(pyridin-4-yl)benzamide | CHEMB...)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human PPARdelta expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor delta(Homo sapiens (Human))TBA

PNG

BDBM50610167(CHEMBL5271038)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human PPARdelta expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor delta(Homo sapiens (Human))TBA

PNG

BDBM50610163(CHEMBL5267263)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human PPARdelta expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor alpha(Homo sapiens (Human))TBA

PNG

BDBM50610167(CHEMBL5271038)

IC50: >5.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional activation preincubated for 6 hrs f...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor alpha(Homo sapiens (Human))TBA

PNG

BDBM50610163(CHEMBL5267263)

IC50: >5.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional activation preincubated for 6 hrs f...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610156(CHEMBL5282748)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610153(CHEMBL5287514)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610150(CHEMBL5281604)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Thyroid hormone receptor beta(Homo sapiens (Human))TBA

PNG

BDBM50610167(CHEMBL5271038)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human THRB expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for 6 hr...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610146(CHEMBL5273188)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610144(CHEMBL5286808)

IC50: >5.00E+3nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610155(CHEMBL5287866)

IC50: 5.25E+3nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))TBA

PNG

BDBM50610157(CHEMBL5273751)

IC50: 7.40E+3nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair

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