Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity at 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 114nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 119nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 163nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 164nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 172nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 245nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 402nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 409nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 462nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 481nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 482nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 928nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.01E+3nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.22E+3nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.27E+3nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.28E+3nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.37E+3nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.49E+3nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.51E+3nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.89E+3nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.49E+3nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Affinity DataKd: 320nMAssay Description:Stabilization of wild type human transthyretin expressed in Escherichia coli BL21(DE3) Star assessed as dissociation constant for TTR-amyloid beta (1...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Affinity DataKd: 810nMAssay Description:Stabilization of wild type human transthyretin expressed in Escherichia coli BL21(DE3) Star assessed as dissociation constant for TTR-amyloid beta (1...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Affinity DataKd: 2.80E+3nMAssay Description:Stabilization of wild type human transthyretin expressed in Escherichia coli BL21(DE3) Star assessed as dissociation constant for TTR-amyloid beta (1...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Affinity DataKd: 1.05E+3nMAssay Description:Stabilization of wild type human transthyretin expressed in Escherichia coli BL21(DE3) Star assessed as dissociation constant for TTR-amyloid beta (1...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Affinity DataKd: 2.70E+3nMAssay Description:Stabilization of wild type human transthyretin expressed in Escherichia coli BL21(DE3) Star assessed as dissociation constant for TTR-amyloid beta (1...More data for this Ligand-Target Pair
TargetGuanylate cyclase soluble subunit alpha-1/beta-1(Homo sapiens (Human))
Baylor University
Curated by ChEMBL
Baylor University
Curated by ChEMBL
Affinity DataEC50: 1.19E+5nMAssay Description:Activation of full length human sGC alpha1/beta1 subunit containing heme in ferric state expressed in Sf9 insect cells using cGMP as substrate incuba...More data for this Ligand-Target Pair
TargetGuanylate cyclase soluble subunit alpha-1/beta-1(Homo sapiens (Human))
Baylor University
Curated by ChEMBL
Baylor University
Curated by ChEMBL
Affinity DataEC50: 1.28E+5nMAssay Description:Activation of full length human sGC alpha1/beta1 subunit containing heme in ferric state expressed in Sf9 insect cells using cGMP as substrate incuba...More data for this Ligand-Target Pair
TargetGuanylate cyclase soluble subunit alpha-1/beta-1(Homo sapiens (Human))
Baylor University
Curated by ChEMBL
Baylor University
Curated by ChEMBL
Affinity DataEC50: 7.07E+5nMAssay Description:Activation of full length human sGC alpha1/beta1 subunit containing heme in ferric state expressed in Sf9 insect cells using cGMP as substrate incuba...More data for this Ligand-Target Pair
TargetGuanylate cyclase soluble subunit alpha-1/beta-1(Homo sapiens (Human))
Baylor University
Curated by ChEMBL
Baylor University
Curated by ChEMBL
Affinity DataEC50: 3.89E+5nMAssay Description:Activation of full length human sGC alpha1/beta1 subunit containing heme in ferric state expressed in Sf9 insect cells using cGMP as substrate incuba...More data for this Ligand-Target Pair
TargetGuanylate cyclase soluble subunit alpha-1/beta-1(Homo sapiens (Human))
Baylor University
Curated by ChEMBL
Baylor University
Curated by ChEMBL
Affinity DataEC50: 5.00E+4nMAssay Description:Activation of full length human sGC alpha1/beta1 subunit containing heme in ferric state expressed in Sf9 insect cells using cGMP as substrate incuba...More data for this Ligand-Target Pair
TargetGuanylate cyclase soluble subunit alpha-1/beta-1(Homo sapiens (Human))
Baylor University
Curated by ChEMBL
Baylor University
Curated by ChEMBL
Affinity DataEC50: 1.66E+5nMAssay Description:Activation of full length human sGC alpha1/beta1 subunit containing heme in ferric state expressed in Sf9 insect cells using cGMP as substrate incuba...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Binding affinity to recombinant human transthyretin expressed in Escherichia coli BL21 by STD-NMR spectroscopic methodMore data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Curated by ChEMBL
Affinity DataKd: 400nMAssay Description:Binding affinity to recombinant human transthyretin expressed in Escherichia coli BL21 by STD-NMR spectroscopic methodMore data for this Ligand-Target Pair