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Found 352 with Last Name = 'hu' and Initial = 'lh'
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM254603(US10214477, Example 5 | US9469597, 4 | US9670136, ...)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50323919(4-(4-(3-(3-tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)ur...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human recombinant full-length N-terminal GST-tagged p38alpha expressed in Escherichia coli by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50323917(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(4-(2-mor...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human recombinant full-length N-terminal GST-tagged p38alpha expressed in Escherichia coli by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of MAO-A (unknown origin)More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM195608(CPI-455)
Affinity DataIC50:  3nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM50481823(CHEMBL5285949)
Affinity DataIC50:  4nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant full-length N-terminal GST-tagged p38alpha expressed in Escherichia coli by radiometric kinase assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM191598(2-(((2-((2-(dimethylamino)ethyl)(ethyl)amino)-2-ox...)
Affinity DataIC50:  4nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM50481825(CHEMBL5277258)
Affinity DataIC50:  7nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase ABL1(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50323918(1-(3-tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)-3-(4-me...)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of mouse recombinant N-terminal His6-tagged Abl by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM50481821(CHEMBL5277129)
Affinity DataIC50:  9nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM50483926(CHEMBL5285505)
Affinity DataIC50:  9nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM50481822(CHEMBL5274997)
Affinity DataIC50:  10nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase ABL1(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataIC50:  10.8nMAssay Description:Inhibition of mouse recombinant N-terminal His6-tagged Abl by radiometric kinase assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50569501(CHEMBL4857832)
Affinity DataIC50:  11nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50308764(4-(3,4-Difluorophenyl)-N-(4-methyl-3-(3-methyl-4-o...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant full length p38alpha assessed as MAPKAPK2 phosphorylation by [32P]ATP SDS-PAGE gel kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50308757(5-(4-Fluorophenyl)-N-(4-methyl-3-(3-methyl-4-oxo-3...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant full length p38alpha assessed as MAPKAPK2 phosphorylation by [32P]ATP SDS-PAGE gel kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM50482594(CHEMBL5290962)
Affinity DataIC50:  17nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50569495(CHEMBL4860694)
Affinity DataIC50:  17nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50323922(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(4-methyl...)
Affinity DataIC50:  18.4nMAssay Description:Inhibition of human recombinant full-length N-terminal GST-tagged p38alpha expressed in Escherichia coli by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))TBA
LigandPNGBDBM26113(2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...)
Affinity DataIC50:  19nMAssay Description:Inhibition of KDM4C (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM223320(KDOAM-25)
Affinity DataIC50:  19nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50569491(CHEMBL4870850)
Affinity DataIC50:  21nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50569489(CHEMBL4851999)
Affinity DataIC50:  24nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50569499(CHEMBL4855257)
Affinity DataIC50:  26nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM195612(GSK467)
Affinity DataIC50:  26nMAssay Description:Inhibition of KDM5B (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50421411(CHEMBL2304168)
Affinity DataIC50:  29nMAssay Description:Compound was evaluated for anti-platelet activating factor potencyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50569500(CHEMBL4871555)
Affinity DataIC50:  35nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  38nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50421412(CHEMBL2304167)
Affinity DataIC50:  40nMAssay Description:Compound was evaluated for anti-platelet activating factor potencyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50569494(CHEMBL4853386)
Affinity DataIC50:  41nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50569493(CHEMBL4855751)
Affinity DataIC50:  42nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50308758(5-(3-Chloro-4-fluorophenyl)-N-(4-methyl-3-(3-methy...)
Affinity DataIC50:  49nMAssay Description:Inhibition of human recombinant full length p38alpha assessed as MAPKAPK2 phosphorylation by [32P]ATP SDS-PAGE gel kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM50481826(CHEMBL5268579)
Affinity DataIC50:  49nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM191599(KDOAM-21 | ethyl 2-(((2-((2-(dimethylamino)ethyl)(...)
Affinity DataIC50:  49nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50421410(CHEMBL2304166)
Affinity DataIC50:  59nMAssay Description:Compound was evaluated for anti-platelet activating factor potencyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50308759(5-(4-Fluoro-3-methylphenyl)-N-(4-methyl-3-(3-methy...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant full length p38alpha assessed as MAPKAPK2 phosphorylation by [32P]ATP SDS-PAGE gel kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase I, thermostable(Thermus aquaticus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123623((R)-13-(3-aminopyrrolidin-1-yl)-12-fluoro-10-oxo-1...)
Affinity DataIC50:  60nMAssay Description:Inhibition of Taq DNA polymeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 6B(Homo sapiens (Human))TBA
LigandPNGBDBM60875(3-((6-(4,5-Dihydro-1H-benzo[d]azepin-3(2H)-yl)-2-(...)
Affinity DataIC50:  60nMAssay Description:Inhibition of KDM6B (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50323919(4-(4-(3-(3-tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)ur...)
Affinity DataIC50:  62.6nMAssay Description:Inhibition of mouse recombinant N-terminal His6-tagged Abl by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM50481827(CHEMBL5269187)
Affinity DataIC50:  65nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50569503(CHEMBL4872523)
Affinity DataIC50:  66nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM15579(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Affinity DataIC50:  70nMAssay Description:Inhibition of MAO-B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  76.2nMAssay Description:Inhibition of human recombinant full-length GST-tagged B-Raf by radiometric kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50:  83.4nMAssay Description:Inhibition of human recombinant full-length GST-tagged B-Raf by radiometric kinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  84nMAssay Description:Inhibition of human recombinant full length p38alpha assessed as MAPKAPK2 phosphorylation by [32P]ATP SDS-PAGE gel kinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  84.8nMAssay Description:Inhibition of human recombinant full-length N-terminal GST-tagged p38alpha expressed in Escherichia coli by radiometric kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50323921(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(4-(2-mor...)
Affinity DataIC50:  92.3nMAssay Description:Inhibition of human recombinant full-length GST-tagged B-Raf by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50308761(CHEMBL591673 | N-(4-Methyl-3-(3-methyl-4-oxo-3,4-d...)
Affinity DataIC50:  94nMAssay Description:Inhibition of human recombinant full length p38alpha assessed as MAPKAPK2 phosphorylation by [32P]ATP SDS-PAGE gel kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50308765(2-tert-Butyl-N-(4-methyl-3-(3-methyl-4-oxo-3,4-dih...)
Affinity DataIC50:  96nMAssay Description:Inhibition of human recombinant full length p38alpha assessed as MAPKAPK2 phosphorylation by [32P]ATP SDS-PAGE gel kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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