Affinity DataKi: 9.10nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Binding Affinity for adenosine A2A receptor expressed in HEK-293 cells compared to [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Binding Affinity for adenosine A2A receptor expressed in HEK-293 cells compared to [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding Affinity for adenosine A2A receptor expressed in HEK-293 cells compared to [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.530nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Inhibition of phosphodiesterase 5 (PDE5) from porcine platelets, range 0.442-0.710More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.730nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.790nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.860nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.930nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.950nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against cyclic AMP production in rat Adenosine A2A receptor assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:50% inhibitory concentration against phosphodiesterase 5 (PDE5) from porcine plateletsMore data for this Ligand-Target Pair