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Found 7 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50006710'
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50006710(8-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50006710(8-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,...)
Affinity DataKi:  7.80nMAssay Description:In vitro binding affinity against Adenosine A2a receptor in rat forebrain membranes by [3H]-NECA (+CPA) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50006710(8-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,...)
Affinity DataKi:  8.5nMAssay Description:Ability to inhibit binding of [3H]-CGS- 21680 to adenosine A2A receptor in rat brain striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50006710(8-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,...)
Affinity DataKi:  42nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50006710(8-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,...)
Affinity DataKi:  42nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50006710(8-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,...)
Affinity DataKi:  71nMAssay Description:Binding Affinity for adenosine A2A receptor expressed in HEK-293 cells compared to [3H]-CGS-21,680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50006710(8-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against cyclic AMP production in rat Adenosine A2A receptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed