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Found 43 with Last Name = 'schwickert' and Initial = 'm'
LigandPNGBDBM50613353(CHEMBL5284517)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of full-length human DNMT2 expressed in bacteria using tRNA-Asp as substrate and 3H-SAM as cosubstrate by tritium incorporation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613356(CHEMBL5273612)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of full-length human DNMT2 expressed in bacteria using tRNA-Asp as substrate and 3H-SAM as cosubstrate by tritium incorporation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613351(CHEMBL5286276)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of full-length human DNMT2 expressed in bacteria using tRNA-Asp as substrate and 3H-SAM as cosubstrate by tritium incorporation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613354(CHEMBL5278294)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of full-length human DNMT2 expressed in bacteria using tRNA-Asp as substrate and 3H-SAM as cosubstrate by tritium incorporation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613350(CHEMBL5285928)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of full-length human DNMT2 expressed in bacteria using tRNA-Asp as substrate and 3H-SAM as cosubstrate by tritium incorporation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613365(CHEMBL5277079)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of human DNMT2 by tritium incorporation assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50597526(CHEMBL5187166)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS by isothermal titration calorimetry ass...More data for this Ligand-Target Pair
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LigandPNGBDBM50378739(SINEFUNGIN | jm2c00120, Sinefungin)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS by isothermal titration calorimetry ass...More data for this Ligand-Target Pair
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LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS by isothermal titration calorimetry ass...More data for this Ligand-Target Pair
LigandPNGBDBM50613355(CHEMBL5273501)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of full-length human DNMT2 expressed in bacteria using tRNA-Asp as substrate and 3H-SAM as cosubstrate by tritium incorporation assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50597525(CHEMBL5202371)
Affinity DataIC50:  3.22E+4nMAssay Description:Inhibition of full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS by isothermal titration calorimetry ass...More data for this Ligand-Target Pair
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LigandPNGBDBM50597524(CHEMBL5173553)
Affinity DataIC50:  3.97E+4nMAssay Description:Inhibition of full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS by isothermal titration calorimetry ass...More data for this Ligand-Target Pair
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LigandPNGBDBM50613352(CHEMBL5272276)
Affinity DataIC50:  6.28E+4nMAssay Description:Inhibition of full-length human DNMT2 expressed in bacteria using tRNA-Asp as substrate and 3H-SAM as cosubstrate by tritium incorporation assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50597523(CHEMBL1091913)
Affinity DataIC50:  7.71E+4nMAssay Description:Inhibition of full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS by isothermal titration calorimetry ass...More data for this Ligand-Target Pair
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LigandPNGBDBM50613351(CHEMBL5286276)
Affinity DataKd:  4.30E+3nMAssay Description:Binding affinity to full-length human DNMT2 expressed in bacteria assessed as apparent dissociation constant by ITC methodMore data for this Ligand-Target Pair
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LigandPNGBDBM50613352(CHEMBL5272276)
Affinity DataKd:  3.21E+4nMAssay Description:Binding affinity to full-length human DNMT2 expressed in bacteria assessed as apparent dissociation constant by ITC methodMore data for this Ligand-Target Pair
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LigandPNGBDBM50613353(CHEMBL5284517)
Affinity DataKd:  1.90E+3nMAssay Description:Binding affinity to full-length human DNMT2 expressed in bacteria assessed as apparent dissociation constant by ITC methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613354(CHEMBL5278294)
Affinity DataKd:  900nMAssay Description:Binding affinity to full-length human DNMT2 expressed in bacteria assessed as apparent dissociation constant by ITC methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50378739(SINEFUNGIN | jm2c00120, Sinefungin)
Affinity DataKd:  2.09E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in Escherichia coli incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50613357(CHEMBL5277756)
Affinity DataKd:  4.51E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50613358(CHEMBL5267824)
Affinity DataKd:  5.58E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613353(CHEMBL5284517)
Affinity DataKd:  2.60E+3nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613359(CHEMBL5272803)
Affinity DataKd:  1.95E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50613360(CHEMBL5270625)
Affinity DataKd:  2.37E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50613361(CHEMBL5279805)
Affinity DataKd:  2.27E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613354(CHEMBL5278294)
Affinity DataKd:  4.20E+3nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613362(CHEMBL5279446)
Affinity DataKd:  1.81E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50613363(CHEMBL5268682)
Affinity DataKd:  1.48E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613350(CHEMBL5285928)
Affinity DataKd:  1.73E+4nMAssay Description:Binding affinity to full-length human DNMT2 expressed in bacteria assessed as apparent dissociation constant by ITC methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50613356(CHEMBL5273612)
Affinity DataKd:  4.90E+3nMAssay Description:Binding affinity to full-length human DNMT2 expressed in bacteria assessed as apparent dissociation constant by ITC methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613355(CHEMBL5273501)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to full-length human DNMT2 expressed in bacteria assessed as apparent dissociation constant by ITC methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613351(CHEMBL5286276)
Affinity DataKd:  2.50E+3nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50613364(CHEMBL5267935)
Affinity DataKd:  1.79E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613350(CHEMBL5285928)
Affinity DataKd:  1.12E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613355(CHEMBL5273501)
Affinity DataKd:  1.04E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613356(CHEMBL5273612)
Affinity DataKd:  2.30E+3nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50597526(CHEMBL5187166)
Affinity DataKd:  8.10E+3nMAssay Description:Binding affinity to full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS assessed as dissociation constant...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50597525(CHEMBL5202371)
Affinity DataKd:  1.05E+4nMAssay Description:Binding affinity to full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS assessed as dissociation constant...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50597524(CHEMBL5173553)
Affinity DataKd:  1.04E+4nMAssay Description:Binding affinity to full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS assessed as dissociation constant...More data for this Ligand-Target Pair
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LigandPNGBDBM50597523(CHEMBL1091913)
Affinity DataKd:  1.14E+4nMAssay Description:Binding affinity to full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS assessed as dissociation constant...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613352(CHEMBL5272276)
Affinity DataKd:  2.82E+4nMAssay Description:Displacement of FTAD from full-length human DNMT2 expressed in bacteria incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
Affinity DataKd:  1.36E+4nMAssay Description:Binding affinity to full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS assessed as dissociation constant...More data for this Ligand-Target Pair
LigandPNGBDBM50378739(SINEFUNGIN | jm2c00120, Sinefungin)
Affinity DataKd:  7.50E+3nMAssay Description:Binding affinity to full length human N-terminal his6-tagged DNMT2 expressed in Escherichia coli Rosetta2(DE3)pLysS assessed as dissociation constant...More data for this Ligand-Target Pair
In DepthDetails PubMed