TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Colorado State University
Curated by ChEMBL
Colorado State University
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Inhibition of human wild type CK2alphaMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Colorado State University
Curated by ChEMBL
Colorado State University
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Inhibition of human wild type CK2alphaMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Colorado State University
Curated by ChEMBL
Colorado State University
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Competitive inhibition of human wild type CK2alpha by Dixon plot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Colorado State University
Curated by ChEMBL
Colorado State University
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Competitive inhibition of human wild type CK2alpha by Dixon plot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Colorado State University
Curated by ChEMBL
Colorado State University
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Competitive inhibition of human wild type CK2alpha by Dixon plot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Colorado State University
Curated by ChEMBL
Colorado State University
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibition of CK2alpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the mouse cerebral cor...More data for this Ligand-Target Pair
Affinity DataIC50: 5.60nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the mouse cerebral cor...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the mouse cerebral cor...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:In vitro Oxytocin receptor antagonistic activity against rat uterine stripsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibitory activity against bovine cathepsin DMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the mouse cerebral cor...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the mouse cerebral cor...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:In vitro inhibitory activity against aspartic proteinases pepsin from porcineMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the mouse cerebral cor...More data for this Ligand-Target Pair
Affinity DataIC50: 85nMAssay Description:In vitro Oxytocin receptor antagonistic activity against rat uterine stripsMore data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the mouse cerebral cor...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 224nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 338nMAssay Description:ETA receptor antagonist activity was measured by inhibition of ET-1 induced vasoconstriction in isolated porcine coronary arteryMore data for this Ligand-Target Pair
Affinity DataIC50: 585nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 680nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the rat pancreas (CCK-...More data for this Ligand-Target Pair
Affinity DataIC50: 690nMAssay Description:In vitro Oxytocin receptor antagonistic activity against rat uterine stripsMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the rat pancreas (CCK-...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 1.07E+3nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the rat pancreas (CCK-...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the rat pancreas (CCK-...More data for this Ligand-Target Pair
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the rat pancreas (CCK-...More data for this Ligand-Target Pair
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 2.47E+3nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:The concentration (nM) producing half-maximal inhibition of specific binding of [1251] Bolton Hunter CCK-8 to CCK receptors in the rat pancreas (CCK-...More data for this Ligand-Target Pair