TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.790nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 820nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.20E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.05E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.20E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences And Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured after 24 hrs by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of phorbol ester-induced ornithine decraboxylase in human MCF7 cells after 6 hrsMore data for this Ligand-Target Pair