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Found 66 with Last Name = 'kelly' and Initial = 'nm'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435322(CHEMBL2391376)
Affinity DataIC50:  180nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435311(CHEMBL2391351)
Affinity DataIC50:  210nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435312(CHEMBL2391354)
Affinity DataIC50:  270nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435314(CHEMBL2391352)
Affinity DataIC50:  390nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435329(CHEMBL2391368)
Affinity DataIC50:  430nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435316(CHEMBL2391382)
Affinity DataIC50:  500nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435340(CHEMBL2391358)
Affinity DataIC50:  590nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435319(CHEMBL2391379)
Affinity DataIC50:  930nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435339(CHEMBL2391359)
Affinity DataIC50:  1.20E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435313(CHEMBL2391353)
Affinity DataIC50:  2.25E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435341(CHEMBL2391357)
Affinity DataIC50:  3.25E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435328(CHEMBL2391369)
Affinity DataIC50:  7.24E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435336(CHEMBL2391362)
Affinity DataIC50:  7.60E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435324(CHEMBL2391374)
Affinity DataIC50:  8.41E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435335(CHEMBL2391363)
Affinity DataIC50:  8.83E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435333(CHEMBL2391365)
Affinity DataIC50:  1.15E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435315(CHEMBL2391539)
Affinity DataIC50:  1.16E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435320(CHEMBL2391378)
Affinity DataIC50:  1.18E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435318(CHEMBL2391380)
Affinity DataIC50:  1.52E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435337(CHEMBL2391361)
Affinity DataIC50:  1.52E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435325(CHEMBL2391373)
Affinity DataIC50:  1.58E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435334(CHEMBL2391364)
Affinity DataIC50:  1.63E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435317(CHEMBL2391381)
Affinity DataIC50:  1.80E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435327(CHEMBL2391371)
Affinity DataIC50:  1.88E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435323(CHEMBL2391375)
Affinity DataIC50:  2.11E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435343(ESAPRAZOLE)
Affinity DataIC50:  2.72E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435326(CHEMBL2391372)
Affinity DataIC50:  8.68E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435342(CHEMBL2391356)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435332(CHEMBL2391366)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435331(CHEMBL2391367)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435330(CHEMBL2391540)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435321(CHEMBL2391377)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research

Curated by ChEMBL
LigandPNGBDBM50435338(CHEMBL2391360)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413340(CHEMBL505715)
Affinity DataEC50:  501nMAssay Description:Agonist activity at human MrgX2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414848(CHEMBL572531)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50394978(CHEMBL573297)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50394977(CHEMBL583068)
Affinity DataEC50:  501nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50394977(CHEMBL583068)
Affinity DataEC50: >3.16E+3nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414849(CHEMBL572766)
Affinity DataEC50:  501nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414850(CHEMBL575058)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414850(CHEMBL575058)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414851(CHEMBL574353)
Affinity DataEC50:  398nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414852(CHEMBL573738)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414852(CHEMBL573738)
Affinity DataEC50:  79.4nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414853(CHEMBL572825)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414853(CHEMBL572825)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414854(CHEMBL574565)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414854(CHEMBL574565)
Affinity DataEC50:  39.8nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414855(CHEMBL573518)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414855(CHEMBL573518)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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