TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 930nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 2.25E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 3.25E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 7.24E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 8.41E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 8.83E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 1.15E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 1.16E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 1.18E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 1.52E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 1.52E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 1.63E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 1.88E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 2.11E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 2.72E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: 8.68E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Nensius Research
Curated by ChEMBL
Nensius Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetMas-related G-protein coupled receptor member X2(Homo sapiens (Human))
Acadia Pharmaceuticals
Curated by ChEMBL
Acadia Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 501nMAssay Description:Agonist activity at human MrgX2 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: >3.16E+3nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 794nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 794nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 79.4nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 39.8nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair