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Found 245 with Last Name = 'frederick' and Initial = 'r'
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50153971(4-(4,6-Dichloro-[1,3,5]triazin-2-ylamino)-benzenes...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50153964(4-((4,6-diethoxy-1,3,5-triazin-2-ylamino)methyl)be...)
Affinity DataKi:  0.340nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50144819(2,3,5,6-Tetrafluoro-N-(3-sulfamoyl-phenyl)-benzami...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(RAT)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333418(7-(4,4,4-Trifluorobutoxy)-1-methyl-beta-carboline ...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333415(7-(Isobutyloxy)-1-methyl-beta-carboline | CHEMBL16...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333419(7-(Cyclohexylmethoxy)-1-methyl-beta-carboline | CH...)
Affinity DataKi:  4.30nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50144825(CHEMBL75620 | N-(2-Bromo-4-sulfamoyl-phenyl)-2,3,5...)
Affinity DataKi:  4.80nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247706(3-(2-amino-3-cyano-1H-pyrrolo[3,2-b]quinoxalin-1-y...)
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333414(7-(Allyloxy)-1-methyl-beta-carboline | CHEMBL16455...)
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333421(7-(Phenethoxy)-1-methyl-beta-carboline | CHEMBL164...)
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247773(4-(3-(4-sulfamoylphenethyl)thioureido)benzoic acid...)
Affinity DataKi:  10nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333420(7-(Benzyloxy)-1-methyl-beta-carboline | CHEMBL1645...)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataKi:  17nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50144819(2,3,5,6-Tetrafluoro-N-(3-sulfamoyl-phenyl)-benzami...)
Affinity DataKi:  21nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM10877(4-(2-hydroxyethyl)benzene-1-sulfonamide | CHEMBL67...)
Affinity DataKi:  22nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  25nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333423(7-(Pyridin-3-ylmethoxy)-1-methyl-beta-carboline | ...)
Affinity DataKi:  25nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333417(2-(1-Methyl-9H-beta-carbolin-7-yloxy)-ethanol | 7-...)
Affinity DataKi:  28nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333416(7-(2-Methoxyethoxy)-1-methyl-beta-carboline | CHEM...)
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50125190(CHEMBL268809 | Quinoline-8-sulfonic acid amide | q...)
Affinity DataKi:  32nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM10861(4-(2-aminoethyl)benzene-1-sulfonamide | CHEMBL7087...)
Affinity DataKi:  33nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333424(7-(Pyridin-4-ylmethoxy)-1-methyl-beta-carboline | ...)
Affinity DataKi:  35nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247720(3-chloro-N-(4-sulfamoylphenethyl)benzo[b]thiophene...)
Affinity DataKi:  51nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247774(1,4-phenylene disulfamate | CHEMBL461964)
Affinity DataKi:  61.6nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50153964(4-((4,6-diethoxy-1,3,5-triazin-2-ylamino)methyl)be...)
Affinity DataKi:  84nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50144825(CHEMBL75620 | N-(2-Bromo-4-sulfamoyl-phenyl)-2,3,5...)
Affinity DataKi:  84nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247760(4-(bis(4-methylpiperidin-1-yl)amino)-N-(4-sulfamoy...)
Affinity DataKi:  90nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333425(7-(Naphthalen-2-ylmethoxy)-1-methyl-beta-carboline...)
Affinity DataKi:  100nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247721(4-fluoro-N-(4-sulfamoylbenzyl)benzenesulfonamide |...)
Affinity DataKi:  100nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50153971(4-(4,6-Dichloro-[1,3,5]triazin-2-ylamino)-benzenes...)
Affinity DataKi:  106nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM10877(4-(2-hydroxyethyl)benzene-1-sulfonamide | CHEMBL67...)
Affinity DataKi:  110nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De Paix

Curated by ChEMBL
LigandPNGBDBM50358044(CHEMBL1917940)
Affinity DataKi:  110nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50125190(CHEMBL268809 | Quinoline-8-sulfonic acid amide | q...)
Affinity DataKi:  125nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De Paix

Curated by ChEMBL
LigandPNGBDBM50358044(CHEMBL1917940)
Affinity DataKi:  160nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells after 1 hr by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM10861(4-(2-aminoethyl)benzene-1-sulfonamide | CHEMBL7087...)
Affinity DataKi:  160nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De Paix

Curated by ChEMBL
LigandPNGBDBM50333419(7-(Cyclohexylmethoxy)-1-methyl-beta-carboline | CH...)
Affinity DataKi:  222nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333428(7-(Ethyloxymorpholine)-1-methyl-beta-carboline | C...)
Affinity DataKi:  256nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247760(4-(bis(4-methylpiperidin-1-yl)amino)-N-(4-sulfamoy...)
Affinity DataKi:  265nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De Paix

Curated by ChEMBL
LigandPNGBDBM50121688(3-Methyl-8-(4,4,4-trifluoro-butoxy)-indeno[1,2-c]p...)
Affinity DataKi:  280nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells after 1 hr by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247719(2-(1,3-dioxoisoindolin-2-yl)-N-(4-sulfamoylpheneth...)
Affinity DataKi:  290nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247721(4-fluoro-N-(4-sulfamoylbenzyl)benzenesulfonamide |...)
Affinity DataKi:  290nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247706(3-(2-amino-3-cyano-1H-pyrrolo[3,2-b]quinoxalin-1-y...)
Affinity DataKi:  300nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247722(2-(3-Allyl-4-oxo-3,4,5,6,7,8-hexahydro-benzo[4,5]t...)
Affinity DataKi:  330nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247773(4-(3-(4-sulfamoylphenethyl)thioureido)benzoic acid...)
Affinity DataKi:  380nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De Paix

Curated by ChEMBL
LigandPNGBDBM50358045(CHEMBL1914652)
Affinity DataKi:  480nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells after 1 hr by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50333422(7-(Pyridin-2-ylmethoxy)-1-methyl-beta-carboline | ...)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus-infected Bacillus thuringiensis israelensis cells after 1 hr by two-step bioluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247774(1,4-phenylene disulfamate | CHEMBL461964)
Affinity DataKi:  643nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50247719(2-(1,3-dioxoisoindolin-2-yl)-N-(4-sulfamoylpheneth...)
Affinity DataKi:  660nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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