TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 8.10nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Binding affinity to FKBP12 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 870nMAssay Description:Binding affinity to FKBP12 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.34E+3nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity to FKBP12 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 2.70E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Binding affinity to FKBP12 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 5.30E+3nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 7.60E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 8.80E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 9.80E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 1.38E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 1.39E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.60E+4nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 1.81E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 2.37E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 2.70E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 2.77E+4nMAssay Description:Binding affinity to FKBP12 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 5.11E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: 6.48E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry
Curated by ChEMBL
Max Institute Of Psychiatry
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair