TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0170nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0200nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0230nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0230nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0280nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0290nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0330nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0330nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0350nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0360nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0360nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0380nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0390nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0430nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0470nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0500nMAssay Description:Binding affinity for dopamine receptor D2 long expressed in Sf9 cells using [125I]-IABN radioligand.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0570nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0580nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Displacement of [125I]ABN from human dopamine D2 long receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Displacement of [125I]IABN from recombinant human D2 long receptor stably expressed in HEK293 cell membranes measured after 60 mins by scintillation ...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0620nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0630nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0630nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0670nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0690nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Displacement of [125I]ABN from human recombinant D2L receptor expressed in HEK cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0700nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0870nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0960nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.118nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.119nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.120nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of (-)-[3H]vesamicol from human VAChT expressed in rat PC12 A123.7 cells after 20 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Displacement of [125I]ABN from human recombinant D2L receptor expressed in HEK cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:In vitro binding affinity on D3 receptor is inhibition of binding of [125I]- NCQ 298 to Sf9 cells infected with recombinant baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Displacement of 2,3-dimethoxy-5-[125I]-iodo-N-[9-benzyl-9-azabicyclo[3.3.1]nonan-3beta-yl]benzamide from human dopamine D2L receptor expressed in HEK...More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Displacement of [125I]ABN from human D3 receptor transfected in HEK-293 cell membrane after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Displacement of [125]IABN from human D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of 2,3-dimethoxy-5-[125I]-iodo-N-[9-benzyl-9-azabicyclo[3.3.1]nonan-3beta-yl]benzamide from human dopamine D3 receptor expressed in HEK2...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.200nMAssay Description:Binding affinity for dopamine receptor D2 long expressed in Sf9 cells using [125I]-IABN radioligand.More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:In vitro binding affinity on D3 receptor is inhibition of binding of [125I]- NCQ 298 to Sf9 cells infected with recombinant baculovirusMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.213nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair