TargetCytochrome P450 1A2(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin) using midazolam as substrateMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
TargetCytochrome P450 2C19(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
TargetCytochrome P450 2C9(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 8.20nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 3.70nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 3.60nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 4.80nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetMitofusin-2(Homo sapiens)
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human Mitofusin-2 expressed in MEF cells assessed as enhancement of mitochondrial elongation and polarization measured after 48 hrs by ...More data for this Ligand-Target Pair
TargetMitofusin-2(Homo sapiens)
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataEC50: 3.80nMAssay Description:Activation of human Mitofusin-2 expressed in MEF cells assessed as enhancement of mitochondrial elongation and polarization measured after 48 hrs by ...More data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 4.20nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 7.10nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 8.80nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetMitofusin-2(Homo sapiens)
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataEC50: 2.5nMAssay Description:Activation of human Mitofusin-2 expressed in MEF cells assessed as enhancement of mitochondrial elongation and polarization measured after 48 hrs by ...More data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 3.10nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Koneru Lakshmaiah Education Foundation
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells after 24 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair