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Found 92 with Last Name = 'tudhope' and Initial = 'sj'
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235359(CHEMBL4088242)
Affinity DataIC50:  0.800nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235343(CHEMBL4103249)
Affinity DataIC50:  1nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235335(CHEMBL4092981)
Affinity DataIC50:  2nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235348(CHEMBL4078988)
Affinity DataIC50:  3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 14(Homo sapiens (Human))
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50541592(CHEMBL3187788)
Affinity DataIC50:  4nMAssay Description:Inhibition of His6-tagged human NIK (330 to 680 residues) S549D mutant expressed in baculovirus-infected Sf9 cells incubated for 30 mins in presence ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235342(CHEMBL319467 | NU-6102)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235346(CHEMBL4102518)
Affinity DataIC50:  8nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 14(Homo sapiens (Human))
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50457815(CHEMBL4211840)
Affinity DataIC50:  10nMAssay Description:Inhibition of His6-tagged human NIK (330 to 680 residues) S549D mutant expressed in baculovirus-infected Sf9 cells incubated for 30 mins in presence ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235347(CHEMBL4078246)
Affinity DataIC50:  10nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235349(CHEMBL4065402)
Affinity DataIC50:  17nMAssay Description:In vitro inhibition against angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235336(CHEMBL4085238)
Affinity DataIC50:  18nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235344(CHEMBL4086832)
Affinity DataIC50:  19nMAssay Description:In vitro inhibition against angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235354(CHEMBL4069161)
Affinity DataIC50:  19nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235345(CHEMBL4105278)
Affinity DataIC50:  24nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235340(CHEMBL4101626)
Affinity DataIC50:  26nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235337(CHEMBL4062554)
Affinity DataIC50:  26nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235355(CHEMBL4081027)
Affinity DataIC50:  39nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 14(Homo sapiens (Human))
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50429614(CHEMBL2334589)
Affinity DataIC50:  40nMAssay Description:Inhibition of His6-tagged human NIK (330 to 680 residues) S549D mutant expressed in baculovirus-infected Sf9 cells incubated for 30 mins in presence ...More data for this Ligand-Target Pair
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235334(CHEMBL4070391)
Affinity DataIC50:  44nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235356(CHEMBL4097571)
Affinity DataIC50:  52nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235343(CHEMBL4103249)
Affinity DataIC50:  97nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 14(Homo sapiens (Human))
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50601633(CHEMBL5196202)
Affinity DataIC50:  200nMAssay Description:Inhibition of His6-tagged human NIK (330 to 680 residues) S549D mutant expressed in baculovirus-infected Sf9 cells incubated for 30 mins in presence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235353(CHEMBL4090226)
Affinity DataIC50:  220nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235342(CHEMBL319467 | NU-6102)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity was determined against baker's yeast Alpha-GlucosidaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 14(Homo sapiens (Human))
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50601626(CHEMBL5198459)
Affinity DataIC50:  251nMAssay Description:Inhibition of His6-tagged human NIK (330 to 680 residues) S549D mutant expressed in baculovirus-infected Sf9 cells incubated for 30 mins in presence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235332(CHEMBL4094205)
Affinity DataIC50:  290nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 14(Homo sapiens (Human))
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50601631(CHEMBL5175837)
Affinity DataIC50:  316nMAssay Description:Inhibition of His6-tagged human NIK (330 to 680 residues) S549D mutant expressed in baculovirus-infected Sf9 cells incubated for 30 mins in presence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235342(CHEMBL319467 | NU-6102)
Affinity DataIC50:  480nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235343(CHEMBL4103249)
Affinity DataIC50:  570nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235345(CHEMBL4105278)
Affinity DataIC50:  570nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk9/human full-length Cyclin T expressed in baculovirus infected Sf21 insect cell...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235357(CHEMBL4089837)
Affinity DataIC50:  580nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235345(CHEMBL4105278)
Affinity DataIC50:  730nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235335(CHEMBL4092981)
Affinity DataIC50:  750nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk9/human full-length Cyclin T expressed in baculovirus infected Sf21 insect cell...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235335(CHEMBL4092981)
Affinity DataIC50:  750nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235361(CHEMBL4074015)
Affinity DataIC50:  830nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235344(CHEMBL4086832)
Affinity DataIC50:  940nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM5530(2-Anilino-6-cyclohexylmethoxypurine | 6-(cyclohexy...)
Affinity DataIC50:  970nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235337(CHEMBL4062554)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk9/human full-length Cyclin T expressed in baculovirus infected Sf21 insect cell...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235342(CHEMBL319467 | NU-6102)
Affinity DataIC50:  1.07E+3nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235329(CHEMBL4061761)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235339(CHEMBL4073211)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 14(Homo sapiens (Human))
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50601627(CHEMBL5196977)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of His6-tagged human NIK (330 to 680 residues) S549D mutant expressed in baculovirus-infected Sf9 cells incubated for 30 mins in presence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase 14(Homo sapiens (Human))
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50601641(CHEMBL5182375)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of His6-tagged human NIK (330 to 680 residues) S549D mutant expressed in baculovirus-infected Sf9 cells incubated for 30 mins in presence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase 14(Homo sapiens (Human))
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50601632(CHEMBL5170825)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of His6-tagged human NIK (330 to 680 residues) S549D mutant expressed in baculovirus-infected Sf9 cells incubated for 30 mins in presence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235336(CHEMBL4085238)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity was determined against bovine liver beta galactosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235337(CHEMBL4062554)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibitory activity was determined against baker's yeast Alpha-GlucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235343(CHEMBL4103249)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk7/recombinant human full-length Cyclin H expressed in baculovirus infected Sf21...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 14(Homo sapiens (Human))
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50601628(CHEMBL5197109)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of His6-tagged human NIK (330 to 680 residues) S549D mutant expressed in baculovirus-infected Sf9 cells incubated for 30 mins in presence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235335(CHEMBL4092981)
Affinity DataIC50:  3.30E+3nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235337(CHEMBL4062554)
Affinity DataIC50:  4.10E+3nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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