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Found 562 with Last Name = 'cohen' and Initial = 'sm'
TargetLactoylglutathione lyase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50402202(CHEMBL2203964)
Affinity DataKi:  11nMAssay Description:Inhibition of human GLO1More data for this Ligand-Target Pair
TargetLactoylglutathione lyase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50092825(CHEMBL128935 | S-(N-phenyl-N-hydroxycarbamoyl)glut...)
Affinity DataKi:  14nMAssay Description:Inhibition of human GLO1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50517464(CHEMBL1234300)
Affinity DataKi:  230nMAssay Description:Inhibition of human GLO1More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50089657(CHEMBL3577298)
Affinity DataKi:  250nMAssay Description:Binding affinity to human Zn2+-HDAC8 assessed as loss of activity by Fluor-de-Lys activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM23274((2E)-3-(2,4-dichlorophenyl)-N-hydroxyprop-2-enamid...)
Affinity DataKi:  300nMAssay Description:Inhibition of Clostridium botulinum BoNT/A using SNAP-25 (141-206) as substrate by HPLC analysisMore data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546871(CHEMBL4745069)
Affinity DataKi:  2.00E+3nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate preincu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50089657(CHEMBL3577298)
Affinity DataKi:  7.00E+3nMAssay Description:Reversible-time dependent inhibition of human wild type HDAC8 by Fluor-de-Lys activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50048539(CHEMBL3309328)
Affinity DataKi:  7.70E+3nMAssay Description:Irreversible inhibition of recombinant Clostridium botulinum N-terminal 6His-tagged BoNT/A (Met1 to Phe425 residues) catalytic domain expressed in Es...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546870(CHEMBL4790141)
Affinity DataKi:  8.90E+3nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate preincu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50057418(CHEMBL3326435)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546872(CHEMBL4761825)
Affinity DataKi:  1.70E+4nMAssay Description:Time dependent inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate by me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546874(CHEMBL4795025)
Affinity DataKi:  3.20E+4nMAssay Description:Time dependent inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate by me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50057411(CHEMBL3326430)
Affinity DataKi:  3.80E+4nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546876(CHEMBL4787837)
Affinity DataKi:  3.80E+4nMAssay Description:Time dependent inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate by me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546880(CHEMBL4799810)
Affinity DataKi:  4.10E+4nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide as substrate preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50057412(CHEMBL3326429)
Affinity DataKi:  4.80E+4nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546875(CHEMBL4746123)
Affinity DataKi:  4.80E+4nMAssay Description:Time dependent inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate by me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50048539(CHEMBL3309328)
Affinity DataKi:  5.20E+4nMAssay Description:Covalent inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50057406(CHEMBL3326434)
Affinity DataKi:  6.40E+4nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546878(CHEMBL4790780)
Affinity DataKi:  6.60E+4nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide as substrate preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546879(CHEMBL4787587)
Affinity DataKi:  8.80E+4nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide as substrate preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546877(CHEMBL4743480)
Affinity DataKi:  8.80E+4nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate preincu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50057410(CHEMBL3326431)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50057417(CHEMBL3326436)
Affinity DataKi:  2.70E+5nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM60985(1-hydroxy-2-pyridinethione | 1-hydroxypyridine-2-t...)
Affinity DataKi:  5.10E+5nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50057414(CHEMBL3326439)
Affinity DataKi:  9.50E+5nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50057408(CHEMBL3326433)
Affinity DataKi:  9.50E+5nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546881(CHEMBL4761785)
Affinity DataKi:  9.98E+5nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide as substrate preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50057415(CHEMBL3326438)
Affinity DataKi:  2.30E+6nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50057409(CHEMBL3326432)
Affinity DataKi:  2.30E+6nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50057416(CHEMBL3326437)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of human carbonic anhydrase using p-nitrophenylacetate as substrate preincubated for 10 mins before substrate addition by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509165(CHEMBL4459575)
Affinity DataIC50: >2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509155(CHEMBL4440123)
Affinity DataIC50: >2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509159(CHEMBL4588964)
Affinity DataIC50: >2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509155(CHEMBL4440123)
Affinity DataIC50: <2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509167(CHEMBL4539596)
Affinity DataIC50: >2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509161(CHEMBL4563716)
Affinity DataIC50: >2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509159(CHEMBL4588964)
Affinity DataIC50: <2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509161(CHEMBL4563716)
Affinity DataIC50: <2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509169(CHEMBL4545631)
Affinity DataIC50: >2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509169(CHEMBL4545631)
Affinity DataIC50: <2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509167(CHEMBL4539596)
Affinity DataIC50: <2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509165(CHEMBL4459575)
Affinity DataIC50: <2nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509170(CHEMBL4440338)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509160(CHEMBL4570983)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509170(CHEMBL4440338)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509160(CHEMBL4570983)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509157(CHEMBL4530222)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509157(CHEMBL4530222)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
University of California

Curated by ChEMBL
LigandPNGBDBM50509166(CHEMBL4550646)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of Influenza A virus RNA-dependent RNA polymerase PA N-terminal endonuclease using [6-FAM]AATCGCAGGCAGCACTC[TAM] substrate and measured ov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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