Affinity DataKi: 0.0140nMAssay Description:Displacement of 2-[125I]iodomelatonin from melatonin receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0440nMAssay Description:Displacement of 2-[125I]iodomelatonin from melatonin receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibitory constant of the compound against human thrombin was determined in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibitory constant of the compound against human thrombin was determined in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT1 receptor expressed in CHO cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT2 receptor expressed in COS7 cells incubated for 1.5 hrs by gamma counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Binding affinity to MT2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT2 receptor expressed in CHO cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity to MT2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT2 receptor expressed in NIH3T3 cells membranes by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibitory constant of the compound against human thrombin was determined in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibitory constant of the compound against human thrombin was determined in vitroMore data for this Ligand-Target Pair
Affinity DataKi: 0.204nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT1 receptor expressed in NIH3T3 cells membranes incubated for 90 mins by Cheng-Prusoff equation an...More data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Displacement of 2-[125I]iodomelatonin from melatonin receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT2 receptor expressed in COS7 cells incubated for 1.5 hrs by gamma counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.302nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT2 receptor expressed in NIH3T3 cells membranes incubated for 90 mins by Cheng-Prusoff equation an...More data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT2 receptor expressed in NIH3T3 cells membranes by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.378nMAssay Description:Displacement of 2-[125I]iodomelatonin from chick brain melatonin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibitory constant of the compound against human thrombin was determined in vitro.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataKi: 0.430nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT1 receptor expressed in CHO cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibitory constant of the compound against human thrombin was determined in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Displacement of 2-[125I]iodomelatonin from chick brain melatonin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:Displacement of 2-[125I]iodomelatonin from melatonin receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT1 receptor expressed in NIH3T3 cells membranes by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibitory constant of the compound against human thrombin was determined in vitro.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataKi: 0.820nMAssay Description:Binding affinity to PPARdelta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.880nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT1 receptor expressed in COS7 cells incubated for 1.5 hrs by gamma counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.880nMAssay Description:Binding affinity to MT1 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibitory constant of the compound against human thrombin was determined in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT2 receptor expressed in CHO cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET-based competitive binding assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to PPARgamma (unknown origin) assessed as inhibition constant by Lanthascreen TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity to PPARalpha (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT1 receptor expressed in NIH3T3 cells membranes incubated for 90 mins by Cheng-Prusoff equation an...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibitory constant of the compound against human thrombin was determined in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory constant of the compound against human thrombin was determined in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Displacement of 2-[1251]-iodomelatonin from human MT1 receptor expressed in NIH3T3 cells membranes by radioligand binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Harbin Institute Of Technology
Curated by ChEMBL
Harbin Institute Of Technology
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair