TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human cytomegalovirus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 d...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human cytomegalovirus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 d...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 7.80nMAssay Description:Inhibition of Varicella-Zoster virus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 ...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 8.5nMAssay Description:Inhibition of Varicella-Zoster virus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 ...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 8.80nMAssay Description:Inhibition of human delta DNA polymerase (95 uL) activity in a solution containg 6.4 mM HEPES (pH 7.5) upon incubation for 12 minutes at 26 degrees C...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of human alpha DNA polymerase (95 uL) activity in a solution containg 6.4 mM HEPES (pH 7.5) upon incubation for 12 minutes at 26 degrees C...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of human alpha DNA polymerase (95 uL) activity in a solution containg 6.4 mM HEPES (pH 7.5) upon incubation for 12 minutes at 26 degrees C...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of human cytomegalovirus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 d...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of Varicella-Zoster virus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 ...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human cytomegalovirus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 d...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of human delta DNA polymerase (95 uL) activity in a solution containg 6.4 mM HEPES (pH 7.5) upon incubation for 12 minutes at 26 degrees C...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human cytomegalovirus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 d...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of human cytomegalovirus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 d...More data for this Ligand-Target Pair
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.79E+3nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.33E+3nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.92E+3nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.41E+3nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of MetAP2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetCytochrome P450 2C9(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
TargetCytochrome P450 1A2(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
TargetCytochrome P450 2C19(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin) using midazolam as substrateMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
TargetMitofusin-2(Homo sapiens)
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataEC50: 3.80nMAssay Description:Activation of human Mitofusin-2 expressed in MEF cells assessed as enhancement of mitochondrial elongation and polarization measured after 48 hrs by ...More data for this Ligand-Target Pair
TargetMitofusin-2(Homo sapiens)
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human Mitofusin-2 expressed in MEF cells assessed as enhancement of mitochondrial elongation and polarization measured after 48 hrs by ...More data for this Ligand-Target Pair
TargetMitofusin-2(Homo sapiens)
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
The First Affiliated Hospital Of Xi'An Jiao Tong University
Curated by ChEMBL
Affinity DataEC50: 2.5nMAssay Description:Activation of human Mitofusin-2 expressed in MEF cells assessed as enhancement of mitochondrial elongation and polarization measured after 48 hrs by ...More data for this Ligand-Target Pair
![](/img/powered_by_small.gif)