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Found 63 with Last Name = 'nagaoka' and Initial = 'y'
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50571956(CHEMBL4874608)
Affinity DataKi:  2.60E+3nMAssay Description:Competitive inhibition of recombinant human Cdc25B (351 to 380 residues) assessed as hydrolysis of substrate O-methylfluorescein phosphate by Linewea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)
Affinity DataIC50:  6nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)
Affinity DataIC50:  18nMAssay Description:Inhibition of HDAC2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50229194(CHEMBL251819 | N-(2-amino-5-(thiophen-2-yl)phenyl)...)
Affinity DataIC50:  40nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50365501(CHEMBL1957458)
Affinity DataIC50:  50nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50365503(CHEMBL1957463)
Affinity DataIC50:  60nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50365502(CHEMBL1957459)
Affinity DataIC50:  80nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50365505(CHEMBL1957464)
Affinity DataIC50:  100nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Mus musculus)
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594395(CHEMBL5189146)
Affinity DataIC50:  110nMAssay Description:Inhibition of mouse HDAC6 expressed in human HEK-293T cells using fluorescent peptide Ac-KGLGK(Ac)-MCA as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 6(Mus musculus)
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594394(CHEMBL5195750)
Affinity DataIC50:  260nMAssay Description:Inhibition of mouse HDAC6 expressed in human HEK-293T cells using fluorescent peptide Ac-KGLGK(Ac)-MCA as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 6(Mus musculus)
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594401(CHEMBL5192796)
Affinity DataIC50:  260nMAssay Description:Inhibition of mouse HDAC6 expressed in human HEK-293T cells using fluorescent peptide Ac-KGLGK(Ac)-MCA as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 6(Mus musculus)
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594396(CHEMBL5172611)
Affinity DataIC50:  330nMAssay Description:Inhibition of mouse HDAC6 expressed in human HEK-293T cells using fluorescent peptide Ac-KGLGK(Ac)-MCA as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 6(Mus musculus)
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594398(CHEMBL5175813)
Affinity DataIC50:  430nMAssay Description:Inhibition of mouse HDAC6 expressed in human HEK-293T cells using fluorescent peptide Ac-KGLGK(Ac)-MCA as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50229194(CHEMBL251819 | N-(2-amino-5-(thiophen-2-yl)phenyl)...)
Affinity DataIC50:  470nMAssay Description:Inhibition of HDAC2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  480nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  500nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Mus musculus)
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594397(CHEMBL5193136)
Affinity DataIC50:  580nMAssay Description:Inhibition of mouse HDAC6 expressed in human HEK-293T cells using fluorescent peptide Ac-KGLGK(Ac)-MCA as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594395(CHEMBL5189146)
Affinity DataIC50:  660nMAssay Description:Inhibition of human ERG potassium channel by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50365501(CHEMBL1957458)
Affinity DataIC50:  670nMAssay Description:Inhibition of HDAC2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50320762(CHEMBL1164063 | N-(2-Aminophenyl)-4-(((biphenyl-4-...)
Affinity DataIC50:  700nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50365503(CHEMBL1957463)
Affinity DataIC50:  740nMAssay Description:Inhibition of HDAC2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50320761(CHEMBL1163973 | N-(2-Aminophenyl)-4-(((2-hydroxyet...)
Affinity DataIC50:  800nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50320760(CHEMBL1165774 | N-(2-Aminophenyl)-4-((3,3-dimethyl...)
Affinity DataIC50:  800nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50365502(CHEMBL1957459)
Affinity DataIC50:  800nMAssay Description:Inhibition of HDAC2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50365505(CHEMBL1957464)
Affinity DataIC50:  880nMAssay Description:Inhibition of HDAC2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50320757(CHEMBL1165443 | N-(2-aminophenyl)-4-((biphenyl-4-y...)
Affinity DataIC50:  900nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50320754(CHEMBL1163887 | N-(2-aminophenyl)-4-((4-(thiophen-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50320755(CHEMBL1165102 | N-(2-aminophenyl)-4-((benzo[b]thio...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50365504(CHEMBL407420)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50320759(CHEMBL1164440 | N-(2-Aminophenyl)-4-((N-(4-(thioph...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50459720(CHEMBL4210305)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of recombinant human C-terminal FLAG/His-tagged HDAC1 expressed in baculovirus infected Sf9 insect cells using HDAC substrate 3 measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  1.51E+3nMAssay Description:Inhibition of HDAC2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594397(CHEMBL5193136)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human HDAC4 using fluorescent peptide Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 10 mins followed by substrate addition...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594396(CHEMBL5172611)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human HDAC4 using fluorescent peptide Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 10 mins followed by substrate addition...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50320756(CHEMBL1164335 | N-(2-aminophenyl)-4-((3-(thiophen-...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50365504(CHEMBL407420)
Affinity DataIC50:  3.36E+3nMAssay Description:Inhibition of HDAC2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594397(CHEMBL5193136)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of human HDAC1 expressed in human HEK-293T cells using fluorescent peptide RHKKAc as substrate preincubated for 10 mins followed by substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594395(CHEMBL5189146)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of human HDAC4 using fluorescent peptide Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 10 mins followed by substrate addition...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594395(CHEMBL5189146)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of human HDAC1 expressed in human HEK-293T cells using fluorescent peptide RHKKAc as substrate preincubated for 10 mins followed by substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594396(CHEMBL5172611)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of human HDAC1 expressed in human HEK-293T cells using fluorescent peptide RHKKAc as substrate preincubated for 10 mins followed by substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594398(CHEMBL5175813)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human HDAC4 using fluorescent peptide Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 10 mins followed by substrate addition...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50459720(CHEMBL4210305)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of recombinant human C-terminal FLAG-tagged HDAC2 expressed in baculovirus infected Sf9 insect cells using HDAC substrate 3 measured after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594398(CHEMBL5175813)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of human HDAC1 expressed in human HEK-293T cells using fluorescent peptide RHKKAc as substrate preincubated for 10 mins followed by substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 6(Mus musculus)
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594400(CHEMBL5205202)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of mouse HDAC6 expressed in human HEK-293T cells using fluorescent peptide Ac-KGLGK(Ac)-MCA as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594394(CHEMBL5195750)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of human HDAC1 expressed in human HEK-293T cells using fluorescent peptide RHKKAc as substrate preincubated for 10 mins followed by substr...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594401(CHEMBL5192796)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of human HDAC4 using fluorescent peptide Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 10 mins followed by substrate addition...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50320758(CHEMBL1165580 | N-(2-Aminophenyl)-4-((methyl(4-(th...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50594401(CHEMBL5192796)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of human HDAC1 expressed in human HEK-293T cells using fluorescent peptide RHKKAc as substrate preincubated for 10 mins followed by substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50459720(CHEMBL4210305)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human full length C-terminal His-tagged HDAC3/N-terminal GST-tagged human NCOR2 (395 to 489 residues) co-expressed in baculovirus infec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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