Compile Data Set for Download or QSAR
maximum 50k data
Found 165 with Last Name = 'arnold' and Initial = 'mb'
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50060725(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
Affinity DataKi:  0.75nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM85212(CAS_5311260 | LY341495 | NSC_5311260)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065468(2-(4-Chloro-phenoxymethyl)-4-(3-piperidin-1-yl-pro...)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065469(2-Diphenylacetylamino-5-guanidino-pentanoic acid 4...)
Affinity DataKi:  4.60nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177564(CHEMBL380540 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065463(2-(4-Chloro-phenoxymethyl)-4-((S)-3-piperidin-3-yl...)
Affinity DataKi:  6nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177560(CHEMBL206042 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-(...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177560(CHEMBL206042 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-(...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50074749((1R,4R,5S,6R)-4-Amino-2-oxa-bicyclo[3.1.0]hexane-4...)
Affinity DataKi:  6.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065460(2-(4-Chloro-phenoxymethyl)-4-(2-piperidin-4-yl-eth...)
Affinity DataKi:  7nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177563(CHEMBL380855 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177557(CHEMBL380365 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065477(2-(4-Chloro-phenoxymethyl)-4-(3-piperidin-2-yl-pro...)
Affinity DataKi:  16nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177565(CHEMBL380858 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065467(2-(4-Chloro-phenoxymethyl)-4-((S)-3-piperidin-3-yl...)
Affinity DataKi:  17nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065466(2-(4-Chloro-phenoxymethyl)-4-(2-piperidin-3-yl-eth...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065459(2-(4-Chloro-phenoxymethyl)-4-((R)-3-piperidin-3-yl...)
Affinity DataKi:  27nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065479(2-(4-Chloro-phenoxymethyl)-4-(2-piperidin-2-yl-eth...)
Affinity DataKi:  29nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065461(2-(4-Chloro-phenoxymethyl)-4-(3-piperidin-3-yl-pro...)
Affinity DataKi:  30nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065462(2-(4-Chloro-phenoxymethyl)-4-((R)-3-piperidin-3-yl...)
Affinity DataKi:  41nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177561((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamin...)
Affinity DataKi:  41nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065475(2-(4-Chloro-phenoxymethyl)-4-(2-piperidin-1-yl-eth...)
Affinity DataKi:  43nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50034503((1R,2R)-3-((S)-Amino-carboxy-methyl)-cyclopropane-...)
Affinity DataKi:  61nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177558(CHEMBL438432 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  74nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50013055(2-aminopentanedioateglutamate | L-Glutamate | glut...)
Affinity DataKi:  90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177562(CHEMBL206840 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  96nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065465(2-(4-Chloro-phenoxymethyl)-4-methyl-1-(3-piperidin...)
Affinity DataKi:  97nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177559(CHEMBL379352 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-(...)
Affinity DataKi:  107nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177559(CHEMBL379352 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-(...)
Affinity DataKi:  107nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065476(2-(4-Chloro-phenoxymethyl)-4-(3-piperidin-4-yl-pro...)
Affinity DataKi:  152nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50004899((1R,2S)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...)
Affinity DataKi:  334nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065474(2-(4-Chloro-phenoxymethyl)-7-methyl-1-(3-piperidin...)
Affinity DataKi:  400nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177564(CHEMBL380540 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  420nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065481(2-(4-Chloro-phenoxymethyl)-1-(3-piperidin-3-yl-pro...)
Affinity DataKi:  700nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177557(CHEMBL380365 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  910nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177562(CHEMBL206840 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  920nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065471(2-(4-Chloro-phenoxymethyl)-1-(2-piperidin-4-yl-eth...)
Affinity DataKi:  940nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177561((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamin...)
Affinity DataKi:  950nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065472(2-(4-Chloro-phenoxymethyl)-1-(3-piperidin-4-yl-pro...)
Affinity DataKi:  980nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177563(CHEMBL380855 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065483(2-(4-Chloro-phenoxymethyl)-1-(4-piperidin-3-yl-but...)
Affinity DataKi:  1.21E+3nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065473(2-(4-Chloro-phenoxymethyl)-1-(2-piperidin-3-yl-eth...)
Affinity DataKi:  1.28E+3nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065464(2-(4-Chloro-phenoxymethyl)-5-methyl-1-(3-piperidin...)
Affinity DataKi:  1.29E+3nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177558(CHEMBL438432 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177562(CHEMBL206840 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177564(CHEMBL380540 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177565(CHEMBL380858 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50049747((2S,4R)-2-Amino-4-(4,4-diphenyl-butyl)-pentanedioi...)
Affinity DataKi:  2.01E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50060727(2-(4-Chloro-phenoxymethyl)-1-methyl-3-piperidin-1-...)
Affinity DataKi:  2.31E+3nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50052398((2R,4R)-4-aminopyrrolidine-2,4-dicarboxylic acid |...)
Affinity DataKi:  2.73E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Displayed 1 to 50 (of 165 total ) | Next | Last >>
Jump to: