TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human Telomerase activity in cell free system by TRAP assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetTumor necrosis factor receptor superfamily member 5(Homo sapiens (Human))
Institut De Biologie MoléCulaire Et Cellulaire
Curated by ChEMBL
Institut De Biologie MoléCulaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human CD40L:mouse CD8 tail binding to human CD40 by surface plasmon resonance methodMore data for this Ligand-Target Pair
TargetTumor necrosis factor receptor superfamily member 5(Homo sapiens (Human))
Institut De Biologie MoléCulaire Et Cellulaire
Curated by ChEMBL
Institut De Biologie MoléCulaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibition of recombinant human CD40L:mouse CD8 tail binding to human CD40 by surface plasmon resonance methodMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 730nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Istituto Chimico Internazionale Dr. G. Rende
Curated by ChEMBL
Affinity DataIC50: 940nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human Telomerase activity in cell free system by TRAP assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair