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Found 422 with Last Name = 'bourguignon' and Initial = 'jj'
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402454(CHEMBL2208337)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50449636(BRL-43694 | GRANISETRON | Kytril | LY-278584 | San...)
Affinity DataKi:  0.600nMAssay Description:Compound was evaluated for its binding affinity for 5-hydroxytryptamine 3 receptor by measuring displacement [3H]GR-65630 in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402442(CHEMBL2208303)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402459(CHEMBL2208301)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50014407(2-(piperazin-1-yl)quinoline | 2-Piperazin-1-yl-qui...)
Affinity DataKi:  1.40nMAssay Description:Compound was evaluated for its binding affinity for 5-hydroxytryptamine 3 receptor by measuring displacement [3H]GR-65630 in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402449(CHEMBL2208325)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402453(CHEMBL2208338)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  3.20nMAssay Description:Compound was evaluated for its binding affinity for 5-hydroxytryptamine 3 receptor by measuring displacement [3H]GR-65630 in rat cerebral cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM85330(CAS_68647 | NSC_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  3.30nMAssay Description:Compound was evaluated for its binding affinity for 5-hydroxytryptamine 3 receptor by measuring displacement [3H]GR-65630 in rat cerebral cortexMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402453(CHEMBL2208338)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402444(CHEMBL2208319)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402452(CHEMBL2208320)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402451(CHEMBL2208322)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402451(CHEMBL2208322)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402444(CHEMBL2208319)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402457(CHEMBL2208340)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402443(CHEMBL2208299)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402457(CHEMBL2208340)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402458(CHEMBL2208339)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402440(CHEMBL2208305)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402446(CHEMBL2208316)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402447(CHEMBL2208312)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402438(CHEMBL2208307)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM82561(CAS_40796-97-2 | TROPANYL 3,5-DICHLOROBENZOATE | T...)
Affinity DataKi:  54nMAssay Description:Compound was evaluated for its binding affinity for 5-hydroxytryptamine 3 receptor by measuring displacement [3H]GR-65630 in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402441(CHEMBL2208304)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402437(CHEMBL2208294)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402458(CHEMBL2208339)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402449(CHEMBL2208325)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402455(CHEMBL2208334)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402450(CHEMBL2208323)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280583(CHEMBL423832 | N*2*,N*2*-Diethyl-2-methyl-N*1*-(6-...)
Affinity DataKi:  112nMAssay Description:Compound was tested for its affinity for muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402439(CHEMBL2208306)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402442(CHEMBL2208303)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402447(CHEMBL2208312)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402436(CHEMBL2208296)
Affinity DataKi:  136nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402437(CHEMBL2208294)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402440(CHEMBL2208305)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402452(CHEMBL2208320)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402448(CHEMBL2208326)
Affinity DataKi:  167nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402456(CHEMBL2204019)
Affinity DataKi:  198nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402455(CHEMBL2208334)
Affinity DataKi:  206nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402438(CHEMBL2208307)
Affinity DataKi:  208nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402443(CHEMBL2208299)
Affinity DataKi:  227nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402445(CHEMBL2208317)
Affinity DataKi:  273nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM48320(4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-metho...)
Affinity DataKi:  348nMAssay Description:Compound was evaluated for its binding affinity for 5-hydroxytryptamine 3 receptor by measuring displacement [3H]GR-65630 in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402436(CHEMBL2208296)
Affinity DataKi:  378nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402448(CHEMBL2208326)
Affinity DataKi:  417nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402439(CHEMBL2208306)
Affinity DataKi:  424nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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