Affinity DataIC50: 0.150nMAssay Description:Inhibition of human MMP13 catalytic domainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.580nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.780nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.880nMAssay Description:Inhibition of human MMP13 catalytic domainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.54nMAssay Description:Inhibition of human MMP13 catalytic domainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.61nMAssay Description:Inhibition of human MMP13 catalytic domainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 2.69nMAssay Description:Inhibition of human MMP13 catalytic domainMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb
Bristol-Myers Squibb
Affinity DataIC50: 3nMAssay Description:Assays measuring the enzyme-catalyzed phosphorylation of GST-I kappa B alpha were performed. The phosphorylated substrate was detected using a Phosph...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 3.46nMAssay Description:Inhibition of human MMP13 catalytic domainMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Compound was tested for in vitro inhibitory activity against ProthrombinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.24nMAssay Description:Inhibition of human MMP13 catalytic domainMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair