Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to human cloned adrenergic alpha 2C receptor receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in human A549 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity to human 5HT2A receptor expressed in human A549 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]INBMeO from human 5HT2A receptor expressed in human A549 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Binding affinity to dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to human cloned dopamine D5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]spiperone from dopamine D2-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Binding affinity to dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human cloned adrenergic alpha 2B receptor receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]INBMeO from human 5HT2A receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in human A549 cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Purdue University
Curated by PDSP Ki Database
Purdue University
Curated by PDSP Ki Database
Affinity DataKi: 21nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]INBMeO from human 5HT2A receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]INBMeO from human 5HT2A receptor expressed in human A549 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University
Curated by PDSP Ki Database
Purdue University
Curated by PDSP Ki Database
Affinity DataKi: 28nMAssay Description:Displacement of [3H]INBMeO from human 5HT2A receptor expressed in human A549 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity to dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in human A549 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Binding affinity to dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Binding affinity to 5HT6 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Binding affinity to human cloned dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Binding affinity to human cloned dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in human A549 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Displacement of [3H]INBMeO from human 5HT2A receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Displacement of [3H]INBMeO from human 5HT2A receptor expressed in human A549 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity to human cloned adrenergic alpha 2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 189nMAssay Description:Binding affinity to histamine H1 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University
Curated by PDSP Ki Database
Purdue University
Curated by PDSP Ki Database
Affinity DataKi: 231nMAssay Description:Binding affinity to 5HT2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Displacement of [3H]spiperone from dopamine D2-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 288nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 302nMAssay Description:Binding affinity to dopamine D2 receptorMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Purdue University
Curated by PDSP Ki Database
Purdue University
Curated by PDSP Ki Database
Affinity DataKi: 330nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Displacement of [3H]spiperone from dopamine D2-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Binding affinity to human cloned dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Binding affinity to dopamine D2 receptorMore data for this Ligand-Target Pair