TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-N-methylspiperone from human dopamine D2long receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:Compound was tested for inhibitory activity against the binding of [3H]-spiperone to Dopamine receptor D2 in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-raclopride from recombinant human D2 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting ...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-raclopride from human D2 receptor expressed in HEK cells incubated for 1 hr by Cheng-Prusoff analysis based microbeta scintillat...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 1.80nMAssay Description:Compound was evaluated for binding affinity towards Dopamine receptor D2 in striatal membranes, using [3H]- spiperone as radioligand in the absence o...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:In vitro binding affinity against Dopamine D2 receptor in rat striatal tissue.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Binding affinity against dopamine D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 2.20nMAssay Description:Compound was evaluated for binding affinity towards dopamine receptor D2 in striatal membranes, using [3H]- spiperone as radioligand in the presence ...More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]-methylspiperone from human D2 receptor transfected in CHO-K1 cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 3nMAssay Description:Compound was evaluated for the binding affinity against [3H]U-86,170-labeled D2 sites in cloned CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 3nMAssay Description:Compound was evaluated for the binding affinity against [3H]-U-86,170-labeled dopamine receptor D2 in cloned CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.06nMAssay Description:Displacement of [3H]spiperone from human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]spiperone binding to Dopamine receptor D2 at 0.02 nMMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 7.80nMAssay Description:Binding affinity towards dopamine receptor D2 by displacing [3H]spiperone radioligand in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]spiperone from dopamine D2-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 10nMAssay Description:In vitro binding affinity for dopamine receptor D2 of rat nucleus accumbens labeled with [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]spiperone from human dopamine D2 receptor short form expressed in CHO cellsMore data for this Ligand-Target Pair