Found 317 with Last Name = 'cochet' and Initial = 'c' 
Affinity DataKi: 180nMAssay Description:Competitive inhibition of recombinant human GST-tagged CK2alpha by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKi: 180nMAssay Description:Competitive inhibition of recombinant human GST-tagged CK2alpha by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of N-terminal GST-tagged human CLK2 (138 to end residues) using SR-rich substrate and [gamma-33P]ATP incubated for 40 mins by scintillatio...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human CLK2 in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human CLK2 in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of N-terminal GST-tagged human CLK2 (138 to end residues) using SR-rich substrate and [gamma-33P]ATP incubated for 40 mins by scintillatio...More data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 6.40nMAssay Description:Inhibition of human recombinant DyrK1b by fluorescence-based immunoassayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 6.40nMAssay Description:Inhibition of recombinant human DYRK1B in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 6.40nMAssay Description:Inhibition of human recombinant DyrK1b by fluorescence-based immunoassayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 6.40nMAssay Description:Inhibition of recombinant human DYRK1B in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human recombinant DyrK1a by fluorescence-based immunoassayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human recombinant DyrK1a by fluorescence-based immunoassayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of recombinant human DYRK1A in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of recombinant human DYRK1A in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of rat DYRK1A isolated from brain using KKISGRLSPIMTEQ as substrate and [gamma33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate and [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate and [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant GST-tagged DYRK1B expressed in Escherichia coli using GRSRSRSRSRSR as substrate and [gamma33P]ATP after 30 mins by sc...More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of rat DYRK1A isolated from brain using KKISGRLSPIMTEQ as substrate and [gamma33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of rat recombinant C-terminal truncated GST-tagged DYRK1A expressed in Escherichia coli using GRSRSRSRSRSR as substrate and [gamma33P]ATP ...More data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of human recombinant GST-tagged DYRK1B expressed in Escherichia coli using GRSRSRSRSRSR as substrate and [gamma33P]ATP after 30 mins by sc...More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
