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Found 857 with Last Name = 'costante' and Initial = 'r'
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428089(CHEMBL2323577)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]Deltorphin from DOR in Sprague-Dawley rat brain membrane after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428089(CHEMBL2323577)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]DAMGO from MOR in Sprague-Dawley rat brain membrane after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21014((2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]DAMGO from MOR in Sprague-Dawley rat brain membrane after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087065(4-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]Ile5,6deltorphin-2 from delta opioid receptor in Wistar rat brain membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50026764(CHEMBL3331509)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]Ile5,6deltorphin II from delta opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116436(CHEMBL3604416)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50026762(CHEMBL3331510)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21014((2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]Deltorphin from DOR in Sprague-Dawley rat brain membrane after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116389(CHEMBL3604509)
Affinity DataKi:  2.60nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21014((2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50026762(CHEMBL3331510)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]Ile5,6deltorphin II from delta opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116443(CHEMBL3604409)
Affinity DataKi:  8.80nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116441(CHEMBL3604411)
Affinity DataKi:  8.90nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116440(CHEMBL3604412)
Affinity DataKi:  9.10nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116442(CHEMBL3604410)
Affinity DataKi:  9.60nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116444(CHEMBL3604408)
Affinity DataKi:  11nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116437(CHEMBL3604415)
Affinity DataKi:  11nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116390(CHEMBL3604420)
Affinity DataKi:  12nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116388(CHEMBL3604510)
Affinity DataKi:  12nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116386(CHEMBL3604511)
Affinity DataKi:  12nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116365(CHEMBL3604512)
Affinity DataKi:  12nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116364(CHEMBL3604513)
Affinity DataKi:  12nMAssay Description:Inhibition of human carbonic anhydrase-12 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of human carbonic anhydrase-2 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116389(CHEMBL3604509)
Affinity DataKi:  13nMAssay Description:Inhibition of human carbonic anhydrase-2 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116435(CHEMBL3604417)
Affinity DataKi:  15nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21014((2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]Ile5,6deltorphin II from delta opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116436(CHEMBL3604416)
Affinity DataKi:  16nMAssay Description:Inhibition of human carbonic anhydrase-2 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116362(CHEMBL3604515)
Affinity DataKi:  20nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116364(CHEMBL3604513)
Affinity DataKi:  20nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116388(CHEMBL3604510)
Affinity DataKi:  21nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116361(CHEMBL3604404)
Affinity DataKi:  22nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116386(CHEMBL3604511)
Affinity DataKi:  23nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116390(CHEMBL3604420)
Affinity DataKi:  23nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  25nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116427(CHEMBL3604419)
Affinity DataKi:  25nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116444(CHEMBL3604408)
Affinity DataKi:  25nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116359(CHEMBL3604406)
Affinity DataKi:  26nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116439(CHEMBL3604413)
Affinity DataKi:  26nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116365(CHEMBL3604512)
Affinity DataKi:  27nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116360(CHEMBL3604405)
Affinity DataKi:  27nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116443(CHEMBL3604409)
Affinity DataKi:  27nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116363(CHEMBL3604514)
Affinity DataKi:  28nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116441(CHEMBL3604411)
Affinity DataKi:  31nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116442(CHEMBL3604410)
Affinity DataKi:  32nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50116440(CHEMBL3604412)
Affinity DataKi:  32nMAssay Description:Inhibition of human carbonic anhydrase-9 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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