TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity to sigma 1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to Alpha2C adrenoceptor receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to Alpha2C adrenoceptor receptorMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataKi: 137nMAssay Description:Binding affinity to DATMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataKi: 149nMAssay Description:Binding affinity to sigma 1 receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataKi: 153nMAssay Description:Binding affinity to sigma 1 receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataKi: 2.28E+3nMAssay Description:Binding affinity to sigma 1 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to Alpha2C adrenoceptor receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to Alpha2C adrenoceptor receptorMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to DATMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity at human P2X7 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity at rat P2X7 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity at mouse P2X7 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of agonist-induced calcium flux by fluoro...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of agonist-induced calcium flux by fluo...More data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of BzATP-induced pore formation flux by...More data for this Ligand-Target Pair
Affinity DataIC50: 156nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in human THP1 cells assessed as inhibition of BzATP-induced IL1beta release by enzym...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced pore formationMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced pore formationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced pore formationMore data for this Ligand-Target Pair