TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.0180nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.0280nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.0350nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.0470nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.0560nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Binding affinity for opioid receptor like type, human Opioid receptor like 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.153nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Binding affinities against Opioid receptor delta 1 of rat brain using [3H]-pClPhe4-DPDPE as radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Binding affinities against delta 2 opioid receptor of rat brain using [3H]Ile5,6-deltorphin II as radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.380nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.385nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.390nMAssay Description:Binding affinities against delta 2 opioid receptor of rat brain using [3H]Ile5,6-deltorphin II as radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.435nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.515nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.535nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.745nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 0.940nMAssay Description:Binding affinities against Opioid receptor delta 1 of rat brain using [3H]-pClPhe4-DPDPE as radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinities against delta 2 opioid receptor of rat brain using [3H]Ile5,6-deltorphin II as radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor mu 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
Affinity DataKi: 102nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor delta 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor mu 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 441nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
Affinity DataKi: 496nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 660nMAssay Description:The binding affinity of the compound was measured using [3H]- DAGO against Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 731nMAssay Description:The binding affinity of the compound was measured using [3H]- DAGO against Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 740nMAssay Description:binding affinities against delta opioid receptor of rat brain using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Opioid receptor delta 1 of rat brain using [3H]-nor BNI as radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinities against delta opioid receptor of rat brain using [3H]-nor BNI as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.06E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.09E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor kappa 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:The binding affinity of the compound was measured using [3H]- DAGO against Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 2.13E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair