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Found 77 with Last Name = 'darula' and Initial = 'z'
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057009((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  0.0180nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057008(4-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  0.0280nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057011((S)-3-[((R)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  0.0300nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057007(4-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  0.0350nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057009((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  0.0470nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057009((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  0.0560nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)
Affinity DataKi:  0.100nMAssay Description:Binding affinity for opioid receptor like type, human Opioid receptor like 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057011((S)-3-[((R)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  0.153nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087064(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi:  0.160nMAssay Description:Binding affinities against Opioid receptor delta 1 of rat brain using [3H]-pClPhe4-DPDPE as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057008(4-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  0.310nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087064(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi:  0.340nMAssay Description:Binding affinities against delta 2 opioid receptor of rat brain using [3H]Ile5,6-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057007(4-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  0.380nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057010((S)-4-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  0.385nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087065(4-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataKi:  0.390nMAssay Description:Binding affinities against delta 2 opioid receptor of rat brain using [3H]Ile5,6-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057012((S)-3-[((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  0.435nMAssay Description:The binding affinity of the compound was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057007(4-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  0.515nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057010((S)-4-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  0.535nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057008(4-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  0.745nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087063(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi:  0.940nMAssay Description:Binding affinities against Opioid receptor delta 1 of rat brain using [3H]-pClPhe4-DPDPE as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087063(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi:  1nMAssay Description:Binding affinities against delta 2 opioid receptor of rat brain using [3H]Ile5,6-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057011((S)-3-[((R)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  1.10nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057012((S)-3-[((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  1.70nMAssay Description:The binding affinity of the compound was measured using [3H]- TIPPsi against Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057012((S)-3-[((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  4nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057010((S)-4-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  5.80nMAssay Description:The binding affinity of the compound was measured using [3H]-naltrindole against Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50094634(CHEMBL140979 | N-(4-Amino-2-methyl-quinolin-6-yl)-...)
Affinity DataKi:  8.20nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121316(Ac-Arg-D-Cha-BTD-D-Arg-D-pClPhe-NH2 | CHEMBL358403)
Affinity DataKi:  34nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121313(Ac-Arg-D-Cha-Qaa-D-Arg-D-pClPhe-NH2 | CHEMBL355931)
Affinity DataKi:  35nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121312(Ac-Arg-D-Cha-I2aa-D-Arg-D-pClPhe-NH2 | CHEMBL26660...)
Affinity DataKi:  44nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121316(Ac-Arg-D-Cha-BTD-D-Arg-D-pClPhe-NH2 | CHEMBL358403)
Affinity DataKi:  53nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121312(Ac-Arg-D-Cha-I2aa-D-Arg-D-pClPhe-NH2 | CHEMBL26660...)
Affinity DataKi:  75nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor mu 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121316(Ac-Arg-D-Cha-BTD-D-Arg-D-pClPhe-NH2 | CHEMBL358403)
Affinity DataKi:  78nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50094634(CHEMBL140979 | N-(4-Amino-2-methyl-quinolin-6-yl)-...)
Affinity DataKi:  102nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121312(Ac-Arg-D-Cha-I2aa-D-Arg-D-pClPhe-NH2 | CHEMBL26660...)
Affinity DataKi:  190nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121316(Ac-Arg-D-Cha-BTD-D-Arg-D-pClPhe-NH2 | CHEMBL358403)
Affinity DataKi:  222nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor delta 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)
Affinity DataKi:  270nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor mu 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121313(Ac-Arg-D-Cha-Qaa-D-Arg-D-pClPhe-NH2 | CHEMBL355931)
Affinity DataKi:  441nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121313(Ac-Arg-D-Cha-Qaa-D-Arg-D-pClPhe-NH2 | CHEMBL355931)
Affinity DataKi:  496nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057011((S)-3-[((R)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  660nMAssay Description:The binding affinity of the compound was measured using [3H]- DAGO against Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057007(4-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  731nMAssay Description:The binding affinity of the compound was measured using [3H]- DAGO against Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087064(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi:  740nMAssay Description:binding affinities against delta opioid receptor of rat brain using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087063(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Opioid receptor delta 1 of rat brain using [3H]-nor BNI as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087064(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinities against delta opioid receptor of rat brain using [3H]-nor BNI as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50094634(CHEMBL140979 | N-(4-Amino-2-methyl-quinolin-6-yl)-...)
Affinity DataKi:  1.06E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121315(Ac-Arg-D-Cha-I9aa-D-Arg-D-pClPhe-NH2 | CHEMBL35621...)
Affinity DataKi:  1.09E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor kappa 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121314(Ac-Arg-D-Cha-Phe-5-tBuPro-D-Arg-D-pClPhe-NH2 | CHE...)
Affinity DataKi:  1.70E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121314(Ac-Arg-D-Cha-Phe-5-tBuPro-D-Arg-D-pClPhe-NH2 | CHE...)
Affinity DataKi:  1.70E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121314(Ac-Arg-D-Cha-Phe-5-tBuPro-D-Arg-D-pClPhe-NH2 | CHE...)
Affinity DataKi:  1.70E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50057008(4-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  1.80E+3nMAssay Description:The binding affinity of the compound was measured using [3H]- DAGO against Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50121315(Ac-Arg-D-Cha-I9aa-D-Arg-D-pClPhe-NH2 | CHEMBL35621...)
Affinity DataKi:  2.13E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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