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Found 5 Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor' and Ligand = 'BDBM50087063'
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087063(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi:  0.940nMAssay Description:Binding affinities against Opioid receptor delta 1 of rat brain using [3H]-pClPhe4-DPDPE as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087063(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi:  1nMAssay Description:Binding affinities against delta 2 opioid receptor of rat brain using [3H]Ile5,6-deltorphin II as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087063(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Opioid receptor delta 1 of rat brain using [3H]-nor BNI as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087063(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi: >1.00E+4nMAssay Description:binding affinities against delta opioid receptor of rat brain using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50087063(4-(2-{2-[(2-Amino-6-hydroxy-1,2,3,4-tetrahydro-nap...)
Affinity DataIC50:  6.57nMAssay Description:Inhibitory concentration for inhibition of electrically induced smooth muscle contractions of MVD (mouse vas deferens) myenteric-plexus-longitudinal ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed