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Found 21 with Last Name = 'decroos' and Initial = 'c'
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM152730(7-Amino-N-hydroxypentanamide (6))
Affinity DataIC50:  68nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM152729(6-Amino-N-hydroxypentanamide (5))
Affinity DataIC50:  130nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM152731(8-Amino-N-hydroxypentanamide (7))
Affinity DataIC50:  150nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM152728(5-Amino-N-hydroxypentanamide (4))
Affinity DataIC50:  170nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM152725((3-azaniumylpropyl)(7,7,7-trifluoro-6-oxoheptyl)az...)
Affinity DataIC50:  260nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 500 nM HDAC8 enzyme, 150 μM Ac-Arg-His-Lys(Ac)-Lys(Ac)-aminomethylcoumarin substrate (BML-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM50438390(CHEMBL2414000)
Affinity DataIC50:  270nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM50438391(CHEMBL2413999)
Affinity DataIC50:  390nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM152731(8-Amino-N-hydroxypentanamide (7))
Affinity DataIC50:  2.20E+3nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 500 nM HDAC8 enzyme, 150 μM Ac-Arg-His-Lys(Ac)-Lys(Ac)-aminomethylcoumarin substrate (BML-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM152730(7-Amino-N-hydroxypentanamide (6))
Affinity DataIC50:  5.30E+3nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 500 nM HDAC8 enzyme, 150 μM Ac-Arg-His-Lys(Ac)-Lys(Ac)-aminomethylcoumarin substrate (BML-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM152726((3-azaniumylpropyl)(5-sulfanylpentyl)azanium (2))
Affinity DataIC50:  1.20E+4nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 500 nM HDAC8 enzyme, 150 μM Ac-Arg-His-Lys(Ac)-Lys(Ac)-aminomethylcoumarin substrate (BML-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM152727((3-azaniumylpropyl)[5-(hydroxycarbamoyl)pentyl]aza...)
Affinity DataIC50:  1.40E+4nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 500 nM HDAC8 enzyme, 150 μM Ac-Arg-His-Lys(Ac)-Lys(Ac)-aminomethylcoumarin substrate (BML-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM152729(6-Amino-N-hydroxypentanamide (5))
Affinity DataIC50:  1.90E+4nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 500 nM HDAC8 enzyme, 150 μM Ac-Arg-His-Lys(Ac)-Lys(Ac)-aminomethylcoumarin substrate (BML-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM50438386(CHEMBL2414004)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM50438389(CHEMBL2414001)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM152728(5-Amino-N-hydroxypentanamide (4))
Affinity DataIC50:  1.20E+5nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 500 nM HDAC8 enzyme, 150 μM Ac-Arg-His-Lys(Ac)-Lys(Ac)-aminomethylcoumarin substrate (BML-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM50405937(CHEMBL173782)
Affinity DataIC50:  1.60E+5nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM50438384(CHEMBL2414006)
Affinity DataIC50:  2.30E+5nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM50438388(CHEMBL2414002)
Affinity DataIC50:  3.80E+5nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM50438393(CHEMBL2414007)
Affinity DataIC50:  1.80E+6nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM50438387(CHEMBL2414003)
Affinity DataIC50:  1.90E+6nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania

LigandPNGBDBM50438385(CHEMBL2414005)
Affinity DataIC50:  1.00E+7nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed