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Found 35 with Last Name = 'el-elimat' and Initial = 't'
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50042034((5Z)-7-Oxozeaenol | 5Z-7-Oxozeaenol | CHEBI:67559 ...)
Affinity DataIC50:  8.10nMAssay Description:Inhibition of TAK1 (unknown origin) expressed in sf9 cells assessed as 32P level incorporation into myelin basic protein incubated for 5 mins at 30 d...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50042034((5Z)-7-Oxozeaenol | 5Z-7-Oxozeaenol | CHEBI:67559 ...)
Affinity DataIC50:  11nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020375(CHEMBL3289785)
Affinity DataIC50:  12nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129131(CHEBI:83275 | Hypothemycin | US10434085, Compound ...)
Affinity DataIC50:  33nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129130(CHEMBL3629241)
Affinity DataIC50:  77nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129129(CHEMBL3629242 | US10434085, Compound 7)
Affinity DataIC50:  360nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129128(CHEMBL3629243 | US10434085, Compound 10)
Affinity DataIC50:  380nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129127(CHEMBL3629244)
Affinity DataIC50:  990nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129126((5E)-7-Oxozeaenol | CHEBI:67558 | CHEMBL1801950 | ...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50347546(CHEMBL1801951 | US10434085, Compound LL-Z164-1)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129125(CHEMBL3629245 | US10434085, Compound 6)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human PDE4B2More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50601437(CHEMBL5207648)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50601435(CHEMBL5204172)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020376(CHEBI:81348 | CHEMBL290932)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129124(CHEMBL3629246 | US10434085, Compound 8)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020377(CHEMBL3289786)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50601436(CHEMBL5186891)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50347544(US10434085, Compound zeaenol | ZEAENOL)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50601433(CHEMBL2152644)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human recombinant PTP1B (1 to 322 residues) expressed in Escherichia coli using pNPP as substrate incubated for 10 mins followed by sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50428912(Betulinan C | CHEMBL2331809)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human PDE4B2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50601434(CHEBI:4041 | CYPERIN | Cyperin)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human recombinant PTP1B (1 to 322 residues) expressed in Escherichia coli using pNPP as substrate incubated for 10 mins followed by sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020378(CHEMBL3289787)
Affinity DataIC50:  1.98E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020379(CHEMBL3289788)
Affinity DataIC50:  2.65E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129086(CHEMBL3629247 | US10434085, Compound dihydrohypoth...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129083(CHEMBL3628303)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129084(CHEMBL3629248)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129085(CHEMBL3334712)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020380(CHEMBL3289789)
Affinity DataIC50:  3.01E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM115127(4,5,7-trihydroxy-9,10-diketo-anthracene-2-carboxyl...)
Affinity DataIC50:  3.06E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50428913(CHEMBL2331810)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of human PDE4B2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50312649(6-chloro-4,5,7-trihydroxy-9,10-dioxo-9,10-dihydroa...)
Affinity DataIC50:  3.78E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50428914(BETULINAN A)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of human PDE4B2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020389(CHEMBL3289790)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed