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Found 35 with Last Name = 'fairweather' and Initial = 'jk'
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375292(CHEMBL407200)
Affinity DataKi:  200nMAssay Description:Inhibition of human platelet heparanase by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375290(CHEMBL279625)
Affinity DataKi:  240nMAssay Description:Inhibition of human platelet heparanase by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375291(CHEMBL439118)
Affinity DataKi:  280nMAssay Description:Inhibition of human platelet heparanase by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375287(CHEMBL260220)
Affinity DataKi:  2.23E+3nMAssay Description:Inhibition of human platelet heparanase by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375287(CHEMBL260220)
Affinity DataKi:  6.83E+4nMAssay Description:Inhibition of human platelet heparanase by uncompetitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374504(CHEMBL258321)
Affinity DataIC50:  240nMAssay Description:Binding affinity at FGF1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375289(CHEMBL258980)
Affinity DataIC50:  250nMAssay Description:Inhibition of human platelet heparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375292(CHEMBL407200)
Affinity DataIC50:  800nMAssay Description:Inhibition of human platelet heparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375290(CHEMBL279625)
Affinity DataIC50:  990nMAssay Description:Inhibition of human platelet heparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375291(CHEMBL439118)
Affinity DataIC50:  1.14E+3nMAssay Description:Inhibition of human platelet heparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375287(CHEMBL260220)
Affinity DataIC50:  1.57E+3nMAssay Description:Inhibition of human platelet heparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179253((2R,3S,4S,5S,6R)-2-{[(2R,3S,4S,5R,6R)-2-{[(2R,3S,4...)
Affinity DataIC50:  1.64E+3nMAssay Description:Inhibitory activity against human platelet heparanase by Microcon ultrafiltration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179254((2R,3S,4S,5S,6R)-2-{[(2R,3S,4S,5R,6R)-2-{[(2R,3S,4...)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibitory activity against human platelet heparanase by Microcon ultrafiltration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179256(6-{5-[(3aS,4S,6aR)-2-oxo-hexahydro-1H-thieno[3,4-d...)
Affinity DataIC50:  1.85E+3nMAssay Description:Inhibitory activity against human platelet heparanase by Microcon ultrafiltration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179255(CHEMBL265885 | N-[(2S,3S,4S,5S,6R)-3-{[(2R,3S,4S,5...)
Affinity DataIC50:  2.02E+3nMAssay Description:Inhibitory activity against human platelet heparanase by Microcon ultrafiltration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375293(CHEMBL1627086)
Affinity DataIC50:  2.69E+3nMAssay Description:Inhibition of human platelet heparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50375288(CHEMBL258894)
Affinity DataIC50:  4.15E+3nMAssay Description:Inhibition of human platelet heparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374509(CHEMBL403403)
Affinity DataIC50:  2.90E+5nMAssay Description:Binding affinity at FGF1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179255(CHEMBL265885 | N-[(2S,3S,4S,5S,6R)-3-{[(2R,3S,4S,5...)
Affinity DataKd:  0.660nMAssay Description:Binding affinity for FGF1 by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 2(Homo sapiens (Human))
Progen Industries

Curated by ChEMBL
LigandPNGBDBM50179255(CHEMBL265885 | N-[(2S,3S,4S,5S,6R)-3-{[(2R,3S,4S,5...)
Affinity DataKd:  112nMAssay Description:Binding affinity for FGF2 by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor A(Homo sapiens (Human))
Progen Industries

Curated by ChEMBL
LigandPNGBDBM50179256(6-{5-[(3aS,4S,6aR)-2-oxo-hexahydro-1H-thieno[3,4-d...)
Affinity DataKd:  7.20nMAssay Description:Binding affinity for VEGF by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179256(6-{5-[(3aS,4S,6aR)-2-oxo-hexahydro-1H-thieno[3,4-d...)
Affinity DataKd:  0.390nMAssay Description:Binding affinity for FGF1 by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor A(Homo sapiens (Human))
Progen Industries

Curated by ChEMBL
LigandPNGBDBM50179254((2R,3S,4S,5S,6R)-2-{[(2R,3S,4S,5R,6R)-2-{[(2R,3S,4...)
Affinity DataKd:  1.70nMAssay Description:Binding affinity for VEGF by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374503(CHEMBL1627089)
Affinity DataKd:  1.40E+6nMAssay Description:Binding affinity at FGF1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 2(Homo sapiens (Human))
Progen Industries

Curated by ChEMBL
LigandPNGBDBM50179256(6-{5-[(3aS,4S,6aR)-2-oxo-hexahydro-1H-thieno[3,4-d...)
Affinity DataKd:  84nMAssay Description:Binding affinity for FGF2 by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374505(CHEMBL1627091)
Affinity DataKd:  7.75E+4nMAssay Description:Binding affinity at FGF1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374506(CHEMBL1627090)
Affinity DataKd:  4.79E+4nMAssay Description:Binding affinity at FGF1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374507(CHEMBL1627093)
Affinity DataKd:  2.33E+5nMAssay Description:Binding affinity at FGF1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374508(CHEMBL1627092)
Affinity DataKd:  2.18E+4nMAssay Description:Binding affinity at FGF1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179254((2R,3S,4S,5S,6R)-2-{[(2R,3S,4S,5R,6R)-2-{[(2R,3S,4...)
Affinity DataKd:  0.120nMAssay Description:Binding affinity for FGF1 by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor A(Homo sapiens (Human))
Progen Industries

Curated by ChEMBL
LigandPNGBDBM50179255(CHEMBL265885 | N-[(2S,3S,4S,5S,6R)-3-{[(2R,3S,4S,5...)
Affinity DataKd:  7.10nMAssay Description:Binding affinity for VEGF by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 2(Homo sapiens (Human))
Progen Industries

Curated by ChEMBL
LigandPNGBDBM50179254((2R,3S,4S,5S,6R)-2-{[(2R,3S,4S,5R,6R)-2-{[(2R,3S,4...)
Affinity DataKd:  86nMAssay Description:Binding affinity for FGF2 by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179253((2R,3S,4S,5S,6R)-2-{[(2R,3S,4S,5R,6R)-2-{[(2R,3S,4...)
Affinity DataKd:  0.144nMAssay Description:Binding affinity for FGF1 by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor A(Homo sapiens (Human))
Progen Industries

Curated by ChEMBL
LigandPNGBDBM50179253((2R,3S,4S,5S,6R)-2-{[(2R,3S,4S,5R,6R)-2-{[(2R,3S,4...)
Affinity DataKd:  1.70nMAssay Description:Binding affinity for VEGF by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor 2(Homo sapiens (Human))
Progen Industries

Curated by ChEMBL
LigandPNGBDBM50179253((2R,3S,4S,5S,6R)-2-{[(2R,3S,4S,5R,6R)-2-{[(2R,3S,4...)
Affinity DataKd:  68nMAssay Description:Binding affinity for FGF2 by BIAcore solution affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed