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Found 450 with Last Name = 'ferorelli' and Initial = 's'
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179280(1-(4-(6-methoxynaphthalen-1-yl)butyl)-4-methylpipe...)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145021(1-Cyclohexyl-4-[4-(1,2,3,4-tetrahydro-naphthalen-1...)
Affinity DataKi:  0.0360nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50299711(4-Cyclohexyl-1-[3-(5-methoxy-1,2,3,4-tetrahydronap...)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H](+)-pentazocine ((+)-[2S-(2R,6R,11R)]-1,2,3,4,5,6-hexahydro-6,11-dimethyl- 3-(3-methyl-2-butenyl)-2,6-methano-3-benzazocine- 8-ol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419549(CHEMBL1929282)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50419548(CHEMBL1929281)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-emopamil from delta(8)-delta(7) sterol isomerase in guinea pig liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50359687(CHEMBL1929279 | CHEMBL1929431)
Affinity DataKi:  0.210nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145029(1-Cyclohexyl-4-(4-naphthalen-1-yl-butyl)-piperazin...)
Affinity DataKi:  0.220nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179257((-)-(R)-1-(4-(6-methoxynaphthalen-1-yl)butyl)-3-me...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50299726(1-cyclohexyl-4-(3-cyclohexylpropyl)piperazine | CH...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H](+)-pentazocine ((+)-[2S-(2R,6R,11R)]-1,2,3,4,5,6-hexahydro-6,11-dimethyl- 3-(3-methyl-2-butenyl)-2,6-methano-3-benzazocine- 8-ol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179262(1-(4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145014(1-Cyclohexyl-4-(5-methoxy-1,2,3,4-tetrahydro-napht...)
Affinity DataKi:  0.310nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179260(1-(3-(6-methoxynaphthalen-1-yl)propyl)-3,3-dimethy...)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179260(1-(3-(6-methoxynaphthalen-1-yl)propyl)-3,3-dimethy...)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145019(1-Cyclohexyl-4-[3-(6-methoxy-1,2,3,4-tetrahydro-na...)
Affinity DataKi:  0.360nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179277(1-(4-(6-methoxynaphthalen-1-yl)butyl)-3,3-dimethyl...)
Affinity DataKi:  0.360nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419548(CHEMBL1929281)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50048866(1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydro-na...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor in guinea pig brain after 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50048866(1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydro-na...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145018(1-Cyclohexyl-4-(5-methoxy-1,2,3,4-tetrahydro-napht...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179269(1-(4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179278((+)-(S)-1-(4-(6-methoxynaphthalen-1-yl)butyl)-2-me...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145016(1-Cyclohexyl-4-[3-(1,2,3,4-tetrahydro-naphthalen-1...)
Affinity DataKi:  0.610nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179263((+)-(S)-1-(4-(6-methoxynaphthalen-1-yl)butyl)-3-me...)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50299710(4-Cyclohexyl-1-[N-(5-methoxy-1,2,3,4-tetrahydronap...)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H](+)-pentazocine ((+)-[2S-(2R,6R,11R)]-1,2,3,4,5,6-hexahydro-6,11-dimethyl- 3-(3-methyl-2-butenyl)-2,6-methano-3-benzazocine- 8-ol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50067013(1-[4-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]-emopamil from delta(8)-delta(7) sterol isomerase in guinea pig liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145024(5-[3-(4-Cyclohexyl-piperazin-1-yl)-propyl]-5,6,7,8...)
Affinity DataKi:  0.690nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219753(1-cyclohexyl-4-[3-(7-methoxynaphthalen-1-yl)propyl...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50419545(CHEMBL1929278)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]-emopamil from delta(8)-delta(7) sterol isomerase in guinea pig liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50170660(CHEMBL190883 | CHEMBL521582 | N,N-dipropyl-2-[4-me...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane without cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179259(1-(4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)...)
Affinity DataKi:  1.01nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419550(CHEMBL1929287)
Affinity DataKi:  1.02nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50170660(CHEMBL190883 | CHEMBL521582 | N,N-dipropyl-2-[4-me...)
Affinity DataKi:  1.03nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50299708(1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronap...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H](+)-pentazocine ((+)-[2S-(2R,6R,11R)]-1,2,3,4,5,6-hexahydro-6,11-dimethyl- 3-(3-methyl-2-butenyl)-2,6-methano-3-benzazocine- 8-ol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50419544(CHEMBL1929277)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-emopamil from delta(8)-delta(7) sterol isomerase in guinea pig liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179271(1-(4-(6-methoxynaphthalen-1-yl)butyl)piperidine | ...)
Affinity DataKi:  1.14nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179281(1-(3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)...)
Affinity DataKi:  1.18nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179266(1-(3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179272((-)-(R)-1-(3-(6-methoxynaphthalen-1-yl)propyl)-3-m...)
Affinity DataKi:  1.35nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179275((-)-(R)-1-(4-(6-methoxynaphthalen-1-yl)butyl)-2-me...)
Affinity DataKi:  1.43nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145020(1-Cyclohexyl-4-[5-(1,2,3,4-tetrahydro-naphthalen-1...)
Affinity DataKi:  1.45nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50299708(1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronap...)
Affinity DataKi:  1.46nMAssay Description:Displacement of [3H](+/-)-emopamil from EBP in Dunkin guinea pig liver membrane by radioreceptor binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179276(1-(3-(6-methoxynaphthalen-1-yl)propyl)-4,4-dimethy...)
Affinity DataKi:  1.47nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179268(1-(3-(6-methoxynaphthalen-1-yl)propyl)-4-methylpip...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145027(1-Cyclohexyl-4-[5-(5-methoxy-1,2,3,4-tetrahydro-na...)
Affinity DataKi:  1.52nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145028(1-Cyclohexyl-4-[4-(5-methoxy-1,2,3,4-tetrahydro-na...)
Affinity DataKi:  1.54nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50419543(CHEMBL1929275)
Affinity DataKi:  1.54nMAssay Description:Displacement of [3H]-emopamil from delta(8)-delta(7) sterol isomerase in guinea pig liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50145022(1-Cyclohexyl-4-[3-(5-methoxy-naphthalen-1-yl)-prop...)
Affinity DataKi:  1.57nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145022(1-Cyclohexyl-4-[3-(5-methoxy-naphthalen-1-yl)-prop...)
Affinity DataKi:  1.57nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145013(1-Cyclohexyl-4-[2-(5-methoxy-1,2,3,4-tetrahydro-na...)
Affinity DataKi:  1.57nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419543(CHEMBL1929275)
Affinity DataKi:  1.75nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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