Compile Data Set for Download or QSAR
maximum 50k data
Found 80 with Last Name = 'garrett' and Initial = 'r'
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50303527((2,2,3,3-Tetramethylcyclopropyl)(1-(4,4,4-trifluor...)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membrane incubated for 1 hr by liquid scintillation spectrophotometric anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor measured after 2 hrs by competitive binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50095155((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]DAMGO from human cloned mu-opioid receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50303527((2,2,3,3-Tetramethylcyclopropyl)(1-(4,4,4-trifluor...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membrane incubated for 1 hr by liquid scintillation spectrophotometric a...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50607249(CHEMBL5219510)
Affinity DataKi:  820nMAssay Description:Displacement of [3H]DAMGO from human cloned mu-opioid receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590554(CHEMBL5183556)
Affinity DataKi:  1.95E+3nMAssay Description:Inhibition of Electrophorus electricus AchE assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590549(CHEMBL5175519)
Affinity DataKi:  3.56E+3nMAssay Description:Inhibition of Electrophorus electricus AchE assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590558(CHEMBL5204385)
Affinity DataKi:  3.81E+3nMAssay Description:Inhibition of Electrophorus electricus AchE assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590552(CHEMBL5170874)
Affinity DataKi:  6.24E+3nMAssay Description:Inhibition of Electrophorus electricus AchE assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505095(CHEMBL4483307)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human KLK7 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505092(CHEMBL4475417)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human KLK5 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505096(CHEMBL4436637)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of trypsin (unknown origin) assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505092(CHEMBL4475417)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of trypsin (unknown origin) assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505096(CHEMBL4436637)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human KLK7 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505095(CHEMBL4483307)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of trypsin (unknown origin) assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505092(CHEMBL4475417)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human KLK7 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505093(CHEMBL4570538)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human KLK7 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505098(CHEMBL4444324)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human KLK7 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505094(CHEMBL4530207)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human KLK7 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590554(CHEMBL5183556)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505096(CHEMBL4436637)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of human KLK5 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505095(CHEMBL4483307)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of human KLK5 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590549(CHEMBL5175519)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590558(CHEMBL5204385)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505093(CHEMBL4570538)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human KLK5 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590553(CHEMBL5194995)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590557(CHEMBL5185822)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505099(CHEMBL4476429)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human KLK7 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590552(CHEMBL5170874)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590556(CHEMBL5181853)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505094(CHEMBL4530207)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human KLK5 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590559(CHEMBL5186170)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590557(CHEMBL5185822)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590559(CHEMBL5186170)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590555(CHEMBL5204223)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505097(CHEMBL4557443)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human KLK7 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505097(CHEMBL4557443)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human KLK5 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590551(CHEMBL5189995)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50505098(CHEMBL4444324)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human KLK5 assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590550(CHEMBL5182677)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590548(CHEMBL5197697)
Affinity DataIC50:  2.64E+4nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590558(CHEMBL5204385)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590556(CHEMBL5181853)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590555(CHEMBL5204223)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590553(CHEMBL5194995)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590552(CHEMBL5170874)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590551(CHEMBL5189995)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590550(CHEMBL5182677)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Displayed 1 to 50 (of 80 total ) | Next | Last >>
Jump to: