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Found 87 with Last Name = 'gavioli' and Initial = 'r'
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)
Affinity DataIC50:  7nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525551(CHEMBL4541448)
Affinity DataIC50:  7nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525569(CHEMBL4584892)
Affinity DataIC50:  12nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525552(CHEMBL4556452)
Affinity DataIC50:  14nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50185156(CHEMBL210439 | Hmb-Val-Gln-Leu-VE)
Affinity DataIC50:  20nMAssay Description:Inhibition of trypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50185159(CHEMBL208162 | Hmb-Phe-Gln-Leu-VE)
Affinity DataIC50:  32nMAssay Description:Inhibition of trypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50185155(CHEMBL207774 | H-Phe-Val-Gln-Leu-VE)
Affinity DataIC50:  42nMAssay Description:Inhibition of trypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50370717(EPOXOMYCIN | Epoxomicin)
Affinity DataIC50:  47nMAssay Description:Inhibition of chymotrypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525557(CHEMBL4449972)
Affinity DataIC50:  56nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50185157(CHEMBL210901 | benzyl (S)-4-methyl-1-((S)-4-methyl...)
Affinity DataIC50:  61nMAssay Description:Inhibition of chymotrypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50185158(CHEMBL210091 | H-Tyr-Val-Gln-Leu-VE)
Affinity DataIC50:  83nMAssay Description:Inhibition of trypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525569(CHEMBL4584892)
Affinity DataIC50:  430nMAssay Description:Inhibition of 20S proteosome beta 2 purified from human HCT116 cells using Boc-LRR-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525552(CHEMBL4556452)
Affinity DataIC50:  430nMAssay Description:Inhibition of 20S proteosome beta 2 purified from human HCT116 cells using Boc-LRR-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525565(CHEMBL4451593)
Affinity DataIC50:  480nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525561(CHEMBL4570264)
Affinity DataIC50:  530nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525565(CHEMBL4451593)
Affinity DataIC50:  560nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525557(CHEMBL4449972)
Affinity DataIC50:  590nMAssay Description:Inhibition of 20S proteosome beta 2 purified from human HCT116 cells using Boc-LRR-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525552(CHEMBL4556452)
Affinity DataIC50:  730nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525547(CHEMBL4587250)
Affinity DataIC50:  770nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525546(CHEMBL4462651)
Affinity DataIC50:  920nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50370717(EPOXOMYCIN | Epoxomicin)
Affinity DataIC50:  980nMAssay Description:Inhibition of trypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525546(CHEMBL4462651)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525546(CHEMBL4462651)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of 20S proteosome beta 2 purified from human HCT116 cells using Boc-LRR-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525563(CHEMBL4588752)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibition of 20S proteosome beta 2 purified from human HCT116 cells using Boc-LRR-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50185159(CHEMBL208162 | Hmb-Phe-Gln-Leu-VE)
Affinity DataIC50:  2.23E+3nMAssay Description:Inhibition of chymotrypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50185157(CHEMBL210901 | benzyl (S)-4-methyl-1-((S)-4-methyl...)
Affinity DataIC50:  2.43E+3nMAssay Description:Inhibition of trypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50185155(CHEMBL207774 | H-Phe-Val-Gln-Leu-VE)
Affinity DataIC50:  4.15E+3nMAssay Description:Inhibition of chymotrypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50185158(CHEMBL210091 | H-Tyr-Val-Gln-Leu-VE)
Affinity DataIC50:  4.32E+3nMAssay Description:Inhibition of chymotrypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)
Affinity DataIC50:  4.59E+3nMAssay Description:Inhibition of 20S proteosome beta 2 purified from human HCT116 cells using Boc-LRR-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525569(CHEMBL4584892)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50185156(CHEMBL210439 | Hmb-Val-Gln-Leu-VE)
Affinity DataIC50:  6.67E+3nMAssay Description:Inhibition of chymotrypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525568(CHEMBL4446481)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525557(CHEMBL4449972)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525554(CHEMBL4551724)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525563(CHEMBL4588752)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525548(CHEMBL4447782)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of 20S proteosome beta 2 purified from human HCT116 cells using Boc-LRR-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525561(CHEMBL4570264)
Affinity DataIC50:  1.78E+4nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525564(CHEMBL4469724)
Affinity DataIC50:  2.04E+4nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525554(CHEMBL4551724)
Affinity DataIC50:  2.15E+4nMAssay Description:Inhibition of 20S proteosome beta 2 purified from human HCT116 cells using Boc-LRR-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525556(CHEMBL4558015)
Affinity DataIC50:  3.06E+4nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525547(CHEMBL4587250)
Affinity DataIC50:  3.89E+4nMAssay Description:Inhibition of 20S proteosome beta 2 purified from human HCT116 cells using Boc-LRR-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525554(CHEMBL4551724)
Affinity DataIC50:  5.01E+4nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525564(CHEMBL4469724)
Affinity DataIC50:  5.02E+4nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525548(CHEMBL4447782)
Affinity DataIC50:  5.11E+4nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525562(CHEMBL4585003)
Affinity DataIC50:  5.16E+4nMAssay Description:Inhibition of 20S proteosome beta 2 purified from human HCT116 cells using Boc-LRR-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525567(CHEMBL4567259)
Affinity DataIC50:  5.32E+4nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525551(CHEMBL4541448)
Affinity DataIC50:  5.75E+4nMAssay Description:Inhibition of 20S proteosome beta 1 purified from human HCT116 cells using Z-LLE-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525553(CHEMBL4534838)
Affinity DataIC50:  5.80E+4nMAssay Description:Inhibition of 20S proteosome beta 2 purified from human HCT116 cells using Boc-LRR-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50525563(CHEMBL4588752)
Affinity DataIC50:  6.33E+4nMAssay Description:Inhibition of 20S proteosome beta 5 purified from human HCT116 cells using Suc-LLVY-AMC as substrate incubated for 30 to 120 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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