Compile Data Set for Download or QSAR
maximum 50k data
Found 144 with Last Name = 'gealageas' and Initial = 'r'
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402454(CHEMBL2208337)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402442(CHEMBL2208303)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402459(CHEMBL2208301)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402453(CHEMBL2208338)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402449(CHEMBL2208325)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402444(CHEMBL2208319)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402453(CHEMBL2208338)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402452(CHEMBL2208320)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402451(CHEMBL2208322)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402451(CHEMBL2208322)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402444(CHEMBL2208319)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402457(CHEMBL2208340)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402443(CHEMBL2208299)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402457(CHEMBL2208340)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402458(CHEMBL2208339)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50462575(CHEMBL4238121)
Affinity DataKi:  29nMAssay Description:Inhibition human FA10a using Boc-LeuGly-Arg-AMC fluorogenic substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402440(CHEMBL2208305)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402446(CHEMBL2208316)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402447(CHEMBL2208312)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50514426(CHEMBL4574713)
Affinity DataKi:  50nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402438(CHEMBL2208307)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402441(CHEMBL2208304)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402437(CHEMBL2208294)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402458(CHEMBL2208339)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402449(CHEMBL2208325)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402455(CHEMBL2208334)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402450(CHEMBL2208323)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402439(CHEMBL2208306)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402442(CHEMBL2208303)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402447(CHEMBL2208312)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402436(CHEMBL2208296)
Affinity DataKi:  136nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402437(CHEMBL2208294)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402440(CHEMBL2208305)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402452(CHEMBL2208320)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402448(CHEMBL2208326)
Affinity DataKi:  167nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402456(CHEMBL2204019)
Affinity DataKi:  198nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402455(CHEMBL2208334)
Affinity DataKi:  206nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402438(CHEMBL2208307)
Affinity DataKi:  208nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402443(CHEMBL2208299)
Affinity DataKi:  227nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402445(CHEMBL2208317)
Affinity DataKi:  273nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402436(CHEMBL2208296)
Affinity DataKi:  378nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402448(CHEMBL2208326)
Affinity DataKi:  417nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402439(CHEMBL2208306)
Affinity DataKi:  424nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402446(CHEMBL2208316)
Affinity DataKi:  425nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402454(CHEMBL2208337)
Affinity DataKi:  590nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50514409(CHEMBL4549938)
Affinity DataKi:  600nMAssay Description:Binding affinity to MBP-tagged recombinant STAT5b-SH2 domain (unknown origin) using carboxyfluoresceine-labeled phosphotyrosine octapeptide incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402450(CHEMBL2208323)
Affinity DataKi:  672nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50514425(CHEMBL4462026)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity to Staphylococcus aureus biotin protein ligaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 144 total ) | Next | Last >>
Jump to: