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Found 227 with Last Name = 'gupte' and Initial = 'a'
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412833(CHEMBL611772)
Affinity DataKi:  0.290nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412824(CHEMBL611766)
Affinity DataKi:  0.320nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412832(CHEMBL612049)
Affinity DataKi:  0.410nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412826(CHEMBL612048)
Affinity DataKi:  0.460nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412819(CHEMBL611785)
Affinity DataKi:  0.480nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412825(CHEMBL609105)
Affinity DataKi:  0.540nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412848(CHEMBL612052)
Affinity DataKi:  0.570nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412821(CHEMBL608839)
Affinity DataKi:  0.590nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412834(CHEMBL611784)
Affinity DataKi:  0.610nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412841(CHEMBL611782)
Affinity DataKi:  0.610nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412847(CHEMBL611775)
Affinity DataKi:  0.630nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM23617((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-{[(4-nitrophe...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to human ENT1 assessed as [3H]uridine uptake by flow cytometryMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM23617((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-{[(4-nitrophe...)
Affinity DataKi:  0.700nMAssay Description:Displacement of SAENTA-fluorescein from human ENT1 in K562 cells after 45 mins by flow cytometryMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM23617((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-{[(4-nitrophe...)
Affinity DataKi:  0.700nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from K562 cell nucleoside transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM23617((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-{[(4-nitrophe...)
Affinity DataKi:  0.708nMAssay Description:Inhibition of human ENT1More data for this Ligand-Target Pair
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412818(CHEMBL609101)
Affinity DataKi:  0.770nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412844(CHEMBL611780)
Affinity DataKi:  0.860nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412846(CHEMBL612041)
Affinity DataKi:  0.880nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412839(CHEMBL611774)
Affinity DataKi:  0.900nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412845(CHEMBL611783)
Affinity DataKi:  0.950nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412820(CHEMBL608842)
Affinity DataKi:  0.950nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412827(CHEMBL611767)
Affinity DataKi:  0.960nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412842(CHEMBL612040)
Affinity DataKi:  1.10nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50222744((2R,3R,4S,5R)-2-(6-(4-nitrobenzylthio)-2-amino-9H-...)
Affinity DataKi:  1.10nMAssay Description:Displacement of SAENTA-fluorescein from human ENT1 in K562 cells after 45 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412831(CHEMBL612037)
Affinity DataKi:  1.30nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412828(CHEMBL608843)
Affinity DataKi:  1.40nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412823(CHEMBL612057)
Affinity DataKi:  1.5nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412843(CHEMBL609100)
Affinity DataKi:  1.5nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412836(CHEMBL608840)
Affinity DataKi:  1.60nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50413751(CHEMBL61773)
Affinity DataKi:  1.78nMAssay Description:Inhibition of human ENT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412835(CHEMBL612051)
Affinity DataKi:  1.90nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50222749(2-fluoro-6-(4-nitrobenzylthio)-9-beta-D-ribofurano...)
Affinity DataKi:  2.10nMAssay Description:Displacement of SAENTA-fluorescein from human ENT1 in K562 cells after 45 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412829(CHEMBL612044)
Affinity DataKi:  2.70nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412838(CHEMBL608838)
Affinity DataKi:  3.10nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412822(CHEMBL611776)
Affinity DataKi:  3.20nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412837(CHEMBL609103)
Affinity DataKi:  3.20nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50366947(BDBM50413737 | CHEMBL512162 | CHEMBL610941)
Affinity DataKi:  3.80nMAssay Description:Inhibition of human ENT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50366947(BDBM50413737 | CHEMBL512162 | CHEMBL610941)
Affinity DataKi:  3.90nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from K562 cell nucleoside transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50413747(CHEMBL61741)
Affinity DataKi:  4.37nMAssay Description:Inhibition of human ENT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50413740(CHEMBL61915)
Affinity DataKi:  4.57nMAssay Description:Inhibition of human ENT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412830(CHEMBL612042)
Affinity DataKi:  5.10nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50412840(CHEMBL612046)
Affinity DataKi:  5.10nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50324670(((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...)
Affinity DataKi:  6.60nMAssay Description:Inhibition of Mycobacterium tuberculosis MbtA expressed in Escherichia coli assessed as ATP-[32P]Ppi exchangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50413744(CHEMBL432688)
Affinity DataKi:  7.08nMAssay Description:Inhibition of human ENT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50411457(CHEMBL1162040)
Affinity DataKi:  7.30nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant MbtA expressed in Escherichia coli by ATP/PPi exchange assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM23620(2-({6-[bis(2-hydroxyethyl)amino]-4,8-bis(piperidin...)
Affinity DataKi:  8.80nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from K562 cell nucleoside transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50366949(BDBM50413728 | CHEMBL418496 | CHEMBL611841)
Affinity DataKi:  9nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from K562 cell nucleoside transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50366949(BDBM50413728 | CHEMBL418496 | CHEMBL611841)
Affinity DataKi:  9.12nMAssay Description:Inhibition of human ENT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50366954(BDBM50413734 | CHEMBL430946 | CHEMBL608592)
Affinity DataKi:  10nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from K562 cell nucleoside transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50222745(2-iodo-6-(4-nitrobenzylthio)-9-beta-D-ribofuranosy...)
Affinity DataKi:  11nMAssay Description:Displacement of SAENTA-fluorescein from human ENT1 in K562 cells after 45 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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