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Found 205 with Last Name = 'hadjipavlou-litina' and Initial = 'd'
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50448214(CHEMBL3120707)
Affinity DataKi:  47nMAssay Description:Noncompetitive inhibition of electric eel AchE using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349614(CHEMBL1808954)
Affinity DataKi:  290nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349611(CHEMBL1808951 | CHEMBL2216905)
Affinity DataKi:  300nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349616(CHEMBL1808956)
Affinity DataKi:  310nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349612(CHEMBL1808952)
Affinity DataKi:  330nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349615(CHEMBL1808955)
Affinity DataKi:  350nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349613(CHEMBL1808953)
Affinity DataKi:  370nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349617(CHEMBL1808957)
Affinity DataKi:  430nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349618(CHEMBL1808958)
Affinity DataKi:  480nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349609(CHEMBL1808949)
Affinity DataKi:  660nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349608(CHEMBL1808948)
Affinity DataKi:  690nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349607(CHEMBL1808947)
Affinity DataKi:  900nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50349610(CHEMBL1808950)
Affinity DataKi:  950nMAssay Description:Inhibition of thrombin using S-2238 as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50274152((2S,9Z)-octadec-9-ene-1,2-diamine dihydrochloride ...)
Affinity DataKi:  2.18E+4nMAssay Description:Inhibition of Sprague-Dawley rat MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50274153((2R,9Z)-octadec-9-ene-1,2-diamine dihydrochloride ...)
Affinity DataKi:  3.90E+4nMAssay Description:Inhibition of Sprague-Dawley rat MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50274151(CHEMBL473249 | hexadecane-1,2-diamine dihydrochlor...)
Affinity DataKi:  5.87E+4nMAssay Description:Inhibition of Sprague-Dawley rat MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50448218(CHEMBL3120710)
Affinity DataIC50:  7nMAssay Description:Inhibition of electric eel AchE using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured for 5 mins by Ellma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM13065(5-(4-chlorophenyl)-1-(4-methoxyphenyl)-3-(trifluor...)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Alexander Technological Education Institute Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50359885(CHEMBL409741)
Affinity DataIC50:  18nMAssay Description:Inhibition of ovine COX1 assessed as PGF2alpha production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  40nMAssay Description:Inhibition of electric eel AchE using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured for 5 mins by Ellma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50448214(CHEMBL3120707)
Affinity DataIC50:  41nMAssay Description:Inhibition of electric eel AchE using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured for 5 mins by Ellma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298593((R)-2-(2-(7-fluoro-1H-indole-2-carboxamido)benzami...)
Affinity DataIC50:  55nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50448216(CHEMBL3120708)
Affinity DataIC50:  65nMAssay Description:Inhibition of electric eel AchE using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured for 5 mins by Ellma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Alexander Technological Education Institute Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant COX-2 assessed as PGF2alpha production by enzyme immunoassayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50448219(CHEMBL3120712)
Affinity DataIC50:  103nMAssay Description:Inhibition of electric eel AchE using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured for 5 mins by Ellma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298576((R)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-phe...)
Affinity DataIC50:  106nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298589((R)-2-(2-(5-fluoro-1H-indole-2-carboxamido)benzami...)
Affinity DataIC50:  151nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298592((+/-)-2-(2-(7-fluoro-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  159nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  197nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50448215(CHEMBL3120706)
Affinity DataIC50:  290nMAssay Description:Inhibition of electric eel AchE using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured for 5 mins by Ellma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298591((+/-)-2-(2-(6-fluoro-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  294nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Alexander Technological Education Institute Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50359883(CHEMBL407152)
Affinity DataIC50:  310nMAssay Description:Inhibition of ovine COX1 assessed as PGF2alpha production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Alexander Technological Education Institute Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50359887(CHEMBL259902)
Affinity DataIC50:  310nMAssay Description:Inhibition of ovine COX1 assessed as PGF2alpha production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298588((+/-)-2-(2-(5-fluoro-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  314nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298579((+/-)-2-(2-(1-methyl-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  350nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLipoxygenase(Glycine max)
Iqog, Csic

Curated by ChEMBL
LigandPNGBDBM32020(4-[4-(3,4-dihydroxyphenyl)-2,3-dimethyl-butyl]pyro...)
Affinity DataIC50:  500nMAssay Description:Inhibition of soybean lipoxygenase using sodium linoleate as substrate by UV-based analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Alexander Technological Education Institute Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50359884(CHEMBL409276)
Affinity DataIC50:  510nMAssay Description:Inhibition of ovine COX1 assessed as PGF2alpha production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50448217(CHEMBL3120709)
Affinity DataIC50:  530nMAssay Description:Inhibition of electric eel AchE using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured for 5 mins by Ellma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298583((+/-)-3-phenyl-2-(2-(7-(trifluoromethyl)-1H-indole...)
Affinity DataIC50:  538nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50448220(CHEMBL3120711)
Affinity DataIC50:  550nMAssay Description:Inhibition of electric eel AchE using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured for 5 mins by Ellma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298582((+/-)-2-(2-(7-methyl-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  671nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298595((+/-)-2-(2-(benzofuran-2-carboxamido)benzamido)-3-...)
Affinity DataIC50:  891nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298587((+/-)-2-(2-(4-fluoro-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  937nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298586((+/-)-2-(2-(1-methyl-5-nitro-1H-indole-2-carboxami...)
Affinity DataIC50:  1.11E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298596((+/-)-2-(2-(benzo[b]thiophene-2-carboxamido)benzam...)
Affinity DataIC50:  1.12E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298572((+/-)-3-phenyl-2-(2-(4,5,6,7-tetrahydro-1H-indole-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298584((+/-)-2-(2-(5-chloro-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  1.84E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298577((+/-)-2-(2-(1H-indole-3-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  1.87E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298581((+/-)-2-(2-(3-methyl-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  2.06E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Aristotelian University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50298599((+/-)-2-(2-(1H-indene-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  2.53E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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